Found 8 Enz. Inhib. hit(s) with Target = 'N-terminal Xaa-Pro-Lys N-methyltransferase 1' and Ligand = 'BDBM50542788'
Affinity DataKi: 4.90nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 90 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 120 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence ...More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 30 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 60 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKd: 980nMAssay Description:Binding affinity to NTMT1 (unknown origin) assessed as binding constant Kd1 by ITC assayMore data for this Ligand-Target Pair
Affinity DataKd: 47nMAssay Description:Binding affinity to NTMT1 (unknown origin) assessed as binding constant Kd2 by ITC assayMore data for this Ligand-Target Pair