TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against Alpha-1 adrenergic receptor was determined using [3H]WB-4101 radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor was determined using [ [3H]spiperone radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Binding affinity against sigma receptor using [3H]-( +)-SKF10,047 radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Binding affinity against Dopamine receptor D2 was determined using [ [3H]-spiperone radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 111nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 111nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 116nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 127nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 127nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 147nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Ability to inhibit the binding of [3H]spiroperidol in rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 168nMAssay Description:Affinity for dopamine receptor D2 binding sites by its ability to displace [3H]spiperone from rat striatum.More data for this Ligand-Target Pair