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Found 37 with Last Name = 'stumpfe' and Initial = 'd'
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50077217(CHEMBL3416885)
Affinity DataKi:  1nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50077213(CHEMBL3416860)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50077206(CHEMBL3416861)
Affinity DataKi:  4nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50163460(2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(3-trifluoro...)
Affinity DataKi:  14.1nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50163452(2-Amino-4-(3-fluoro-phenyl)-6-(2-hydroxy-ethylsulf...)
Affinity DataKi:  39.8nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50163453(2-Amino-4-(3-difluoromethoxy-phenyl)-6-(2-hydroxy-...)
Affinity DataKi:  39.8nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50077462(CHEMBL3416859)
Affinity DataKi:  81nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50163462(2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-m-tolyl-pyri...)
Affinity DataKi:  81.3nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50077460(CHEMBL3416864)
Affinity DataKi:  295nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50077454(CHEMBL3416858)
Affinity DataKi:  2.83E+3nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50229708(CHEMBL4069862)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM13066(2-{2-[(2,6-dichlorophenyl)amino]phenyl}acetic acid...)
Affinity DataIC50:  3nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM13066(2-{2-[(2,6-dichlorophenyl)amino]phenyl}acetic acid...)
Affinity DataIC50:  5nMAssay Description:Inhibition of COX2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM5380(2,4-Disubstituted Pyrimidine 2d | N-(3,5-dimethylp...)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50229706(CHEMBL4080549)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50207446(2-(2-(2-chloro-6-fluorophenylamino)-5-methylphenyl...)
Affinity DataIC50:  7nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50229707(CHEMBL4098578)
Affinity DataIC50:  20nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50384799(CHEMBL2037483)
Affinity DataIC50:  20nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50364776(CHEMBL1952141 | CHEMBL1952329)
Affinity DataIC50:  20nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50229705(CHEMBL4103924)
Affinity DataIC50:  25nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50364787(CHEMBL1952107)
Affinity DataIC50:  69nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50364806(CHEMBL1952328)
Affinity DataIC50:  130nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50364792(CHEMBL1952112)
Affinity DataIC50:  155nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50229709(CHEMBL4090855)
Affinity DataIC50:  200nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50229710(CHEMBL4076784)
Affinity DataIC50:  316nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM5400(2,4-Disubstituted Pyrimidine 5b | N-(3,5-dimethylp...)
Affinity DataIC50:  2.39E+3nMAssay Description:Antagonist activity at VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM19828((1R,2R)-2-{[(3-chlorophenyl)sulfanyl]methyl}-N-(cy...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM19817((1R,2R)-N-(cyanomethyl)-2-[(phenylsulfanyl)methyl]...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50207446(2-(2-(2-chloro-6-fluorophenylamino)-5-methylphenyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of COX2More data for this Ligand-Target Pair
TargetProcathepsin L(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM19817((1R,2R)-N-(cyanomethyl)-2-[(phenylsulfanyl)methyl]...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50049661(3''''-Fluoro-4''''-methoxy-[1,1'';2'',1'''']terphe...)
Affinity DataIC50:  7.16E+4nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn

Curated by ChEMBL
LigandPNGBDBM50441097(CHEMBL2430564)
Affinity DataIC50:  8.53E+4nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn

Curated by ChEMBL
LigandPNGBDBM50441098(CHEMBL2430563)
Affinity DataIC50:  9.97E+4nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM19828((1R,2R)-2-{[(3-chlorophenyl)sulfanyl]methyl}-N-(cy...)
Affinity DataIC50:  1.02E+5nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn

Curated by ChEMBL
LigandPNGBDBM50441101(CHEMBL2430571)
Affinity DataIC50:  1.19E+5nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn

Curated by ChEMBL
LigandPNGBDBM50441099(CHEMBL2430574)
Affinity DataIC50:  7.40E+5nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn

Curated by ChEMBL
LigandPNGBDBM50441100(CHEMBL2430572)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed