TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 14.1nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 81.3nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 295nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataKi: 2.83E+3nMAssay Description:Antagonist activity at human vasopressin 1a receptorMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Antagonist activity at VEGFR2More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 155nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:Inhibition of tankyrase-2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.39E+3nMAssay Description:Antagonist activity at VEGFR2More data for this Ligand-Target Pair
TargetProcathepsin L(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of cathepsin LMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of COX2More data for this Ligand-Target Pair
TargetProcathepsin L(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of cathepsin LMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T
Curated by ChEMBL
Affinity DataIC50: 7.16E+4nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn
Curated by ChEMBL
University Hospital Of Bonn
Curated by ChEMBL
Affinity DataIC50: 8.53E+4nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn
Curated by ChEMBL
University Hospital Of Bonn
Curated by ChEMBL
Affinity DataIC50: 9.97E+4nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn
Curated by ChEMBL
University Hospital Of Bonn
Curated by ChEMBL
Affinity DataIC50: 1.19E+5nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn
Curated by ChEMBL
University Hospital Of Bonn
Curated by ChEMBL
Affinity DataIC50: 7.40E+5nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair
TargetDelta-aminolevulinic acid dehydratase(Homo sapiens (Human))
University Hospital Of Bonn
Curated by ChEMBL
University Hospital Of Bonn
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human ALADH after 20 minsMore data for this Ligand-Target Pair