Compile Data Set for Download or QSAR
maximum 50k data
Found 64 with Last Name = 'surleraux' and Initial = 'dl'
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123407(US8741926, 91)
Affinity DataKi:  0.0500nM ΔG°:  -59.8kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123410(US8741926, 82 | US8754106, 82 | US8754106, 91)
Affinity DataKi:  0.0500nMAssay Description:The aim of this in vitro assay was to measure the inhibition of HCV NS3/4A protease complexes by the compounds of the present invention. This assay p...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123413(US8741926, 94 | US8754106, 94)
Affinity DataKi:  0.100nM ΔG°:  -58.0kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123411(US8741926, 56)
Affinity DataKi:  0.100nM ΔG°:  -58.0kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123415(US8741926, 95 | US8754106, 95)
Affinity DataKi:  0.100nM ΔG°:  -58.0kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123415(US8741926, 95 | US8754106, 95)
Affinity DataKi:  0.100nMAssay Description:The aim of this in vitro assay was to measure the inhibition of HCV NS3/4A protease complexes by the compounds of the present invention. This assay p...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123413(US8741926, 94 | US8754106, 94)
Affinity DataKi:  0.100nMAssay Description:The aim of this in vitro assay was to measure the inhibition of HCV NS3/4A protease complexes by the compounds of the present invention. This assay p...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM124106(US8754106, 56)
Affinity DataKi:  0.100nMAssay Description:The aim of this in vitro assay was to measure the inhibition of HCV NS3/4A protease complexes by the compounds of the present invention. This assay p...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123414(US8741926, 48 | US8754106, 48)
Affinity DataKi:  0.25nM ΔG°:  -55.7kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123414(US8741926, 48 | US8754106, 48)
Affinity DataKi:  0.25nMAssay Description:The aim of this in vitro assay was to measure the inhibition of HCV NS3/4A protease complexes by the compounds of the present invention. This assay p...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123412(US8741926, 57 | US8754106, 57)
Affinity DataKi:  0.300nM ΔG°:  -55.3kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123412(US8741926, 57 | US8754106, 57)
Affinity DataKi:  0.300nMAssay Description:The aim of this in vitro assay was to measure the inhibition of HCV NS3/4A protease complexes by the compounds of the present invention. This assay p...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM50336504((2R,3aR,10Z,11aS,12aR,14aR)-N-(cyclopropylsulfonyl...)
Affinity DataKi:  0.5nM ΔG°:  -54.0kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM50336504((2R,3aR,10Z,11aS,12aR,14aR)-N-(cyclopropylsulfonyl...)
Affinity DataKi:  0.5nMAssay Description:The aim of this in vitro assay was to measure the inhibition of HCV NS3/4A protease complexes by the compounds of the present invention. This assay p...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM124105(US8754106, 55)
Affinity DataKi:  5nMAssay Description:The aim of this in vitro assay was to measure the inhibition of HCV NS3/4A protease complexes by the compounds of the present invention. This assay p...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123408(US8741926, 55)
Affinity DataKi:  5nM ΔG°:  -48.2kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123410(US8741926, 82 | US8754106, 82 | US8754106, 91)
Affinity DataKi:  9.40nMAssay Description:The aim of this in vitro assay was to measure the inhibition of HCV NS3/4A protease complexes by the compounds of the present invention. This assay p...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123410(US8741926, 82 | US8754106, 82 | US8754106, 91)
Affinity DataKi:  9.40nM ΔG°:  -46.6kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein(Hepatitis C virus)
Janssen Ireland

US Patent
LigandPNGBDBM123409(US8741926, 81)
Affinity DataKi:  1.00E+3nM ΔG°:  -34.8kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of full-length hepatitis C NS3 protease enzyme was measured essentially as described in Poliakov, 2002 Prot Expression & Purification ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50410310(CHEMBL2079773)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50410311(CHEMBL2068731)
Affinity DataIC50:  50nMAssay Description:Inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422732(CHEMBL424782)
Affinity DataIC50:  112nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422734(CHEMBL368301)
Affinity DataIC50:  178nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422722(CHEMBL360752)
Affinity DataIC50:  186nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422731(CHEMBL425516)
Affinity DataIC50:  209nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422706(CHEMBL367104)
Affinity DataIC50:  219nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422718(CHEMBL177640)
Affinity DataIC50:  257nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422733(CHEMBL414654)
Affinity DataIC50:  355nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422697(CHEMBL362252)
Affinity DataIC50:  372nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422703(CHEMBL366982)
Affinity DataIC50:  380nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422711(CHEMBL360274)
Affinity DataIC50:  417nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422699(CHEMBL369841)
Affinity DataIC50:  417nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422721(CHEMBL177622)
Affinity DataIC50:  427nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422704(CHEMBL177215)
Affinity DataIC50:  427nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422700(CHEMBL177515)
Affinity DataIC50:  427nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422728(CHEMBL424780)
Affinity DataIC50:  437nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422702(CHEMBL174793)
Affinity DataIC50:  501nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422724(CHEMBL177724)
Affinity DataIC50:  562nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422696(CHEMBL174001)
Affinity DataIC50:  562nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422715(CHEMBL177690)
Affinity DataIC50:  562nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422708(CHEMBL177380)
Affinity DataIC50:  631nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422698(CHEMBL368424)
Affinity DataIC50:  676nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422730(CHEMBL177405)
Affinity DataIC50:  776nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422713(CHEMBL177311)
Affinity DataIC50:  813nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422709(CHEMBL174851)
Affinity DataIC50:  1.00E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422705(CHEMBL368509)
Affinity DataIC50:  1.05E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422695(CHEMBL175404)
Affinity DataIC50:  1.41E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422717(CHEMBL175671)
Affinity DataIC50:  1.41E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422727(CHEMBL367945)
Affinity DataIC50:  1.45E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422712(CHEMBL177704)
Affinity DataIC50:  1.59E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 64 total ) | Next | Last >>
Jump to: