Affinity DataIC50: 100nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of ovine COX1-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of ovine COX1 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of human ERG by automated planar patch-clamp systemMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human ERG assessed as decrease in tail current amplitude measured after 5 mins by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of human ERG by automated planar patch-clamp systemMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of human ERG by automated planar patch-clamp systemMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human ERG assessed as decrease in tail current amplitude measured after 5 mins by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 2.54E+3nMAssay Description:Inhibition of human ERG by automated planar patch-clamp systemMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 2.54E+3nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human ERG by automated planar patch-clamp systemMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 2.89E+3nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 2.89E+3nMAssay Description:Inhibition of human ERG by automated planar patch-clamp systemMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human ERG assessed as decrease in tail current amplitude measured after 5 mins by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 3.63E+3nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human ERG assessed as decrease in tail current amplitude measured after 5 mins by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibition of ovine COX2 assessed as inhibition of PGF2alpha production from PGH2 preincubated for 5 mins before arachidonic acid addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ovine COX2-mediated prostaglandin alpha production by enzyme immuno assayMore data for this Ligand-Target Pair