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Found 96 with Last Name = 'van camp' and Initial = 'ja'
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25430(4-(2-hydroxyphenyl)-2-(trifluoromethyl)benzonitril...)
Affinity DataIC50:  0.0200nMAssay Description:Antagonist activity at human AR in MDA-MB453-MMTV-luci cells by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220383(4'-methoxy-3-trifluoromethyl-biphenyl-4-carbonitri...)
Affinity DataIC50:  0.800nMAssay Description:Antagonist activity at human AR in MDA-MB453-MMTV-luci cells by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220379(3,2'-bis-trifluoromethyl-biphenyl-4-carbonitrile |...)
Affinity DataIC50: >1nMAssay Description:Antagonist activity at human AR in MDA-MB453-MMTV-luci cells by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216194(CHEMBL391935 | N-(2-chlorophenethyl)-N-(pyrrolidin...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220389(2'-chloro-3-trifluoromethyl-biphenyl-4-carbonitril...)
Affinity DataIC50:  9.80nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220379(3,2'-bis-trifluoromethyl-biphenyl-4-carbonitrile |...)
Affinity DataIC50:  10.9nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220385(4'-hydroxy-3-trifluoromethyl-biphenyl-4-carbonitri...)
Affinity DataIC50:  11.9nMAssay Description:Antagonist activity at human AR in MDA-MB453-MMTV-luci cells by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220384(2',6'-dimethoxy-3-trifluoromethyl-biphenyl-4-carbo...)
Affinity DataIC50:  14.7nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25428(4-[3-(4-hydroxybutyl)-4,4-dimethyl-2,5-dioxoimidaz...)
Affinity DataIC50:  16nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25432(6-{methyl[(1R)-1-phenylethyl]amino}-4-(trifluorome...)
Affinity DataIC50:  20nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220376(2'-methoxy-3-trifluoromethyl-biphenyl-4-carbonitri...)
Affinity DataIC50:  20.1nMAssay Description:Antagonist activity at human AR in MDA-MB453-MMTV-luci cells by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25434(4-(2-hydroxycyclohexyl)-2-(trifluoromethyl)benzoni...)
Affinity DataIC50:  26nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216201(CHEMBL233987 | N-(2-methoxyphenethyl)-4-(6-aza-bic...)
Affinity DataIC50:  29nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220376(2'-methoxy-3-trifluoromethyl-biphenyl-4-carbonitri...)
Affinity DataIC50:  37nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216180(CHEMBL233799 | N-(2-methoxyphenethyl)-N-(pyrrolidi...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25436(4-[(1R,2R)-2-hydroxycyclohexyl]-2-(trifluoromethyl...)
Affinity DataIC50:  37nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25431(4-(2-hydroxyphenyl)-2-methoxybenzonitrile | diaryl...)
Affinity DataIC50:  37nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25430(4-(2-hydroxyphenyl)-2-(trifluoromethyl)benzonitril...)
Affinity DataIC50:  39.9nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25430(4-(2-hydroxyphenyl)-2-(trifluoromethyl)benzonitril...)
Affinity DataIC50:  39.9nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220383(4'-methoxy-3-trifluoromethyl-biphenyl-4-carbonitri...)
Affinity DataIC50:  56.7nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25437((trifluoromethyl)benzonitrile, 14 | 4-{[(1R,2S)-2-...)
Affinity DataIC50:  60nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220385(4'-hydroxy-3-trifluoromethyl-biphenyl-4-carbonitri...)
Affinity DataIC50:  61.2nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216199(4-(2-aza-bicyclo[2.2.1]heptan-2-ylmethyl)-N-(2-met...)
Affinity DataIC50:  95nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216188(CHEMBL233422 | N-(2-methoxyphenethyl)-4-(((1S,2S)-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220388(3'-methoxy-3-trifluoromethyl-biphenyl-4-carbonitri...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at human AR in MDA-MB453-MMTV-luci cells by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216193(CHEMBL233609 | N-(2-methoxyphenethyl)-4-(((S)-2-(m...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220375(2'-methyl-3-trifluoromethyl-biphenyl-4-carbonitril...)
Affinity DataIC50:  146nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216197(CHEMBL233610 | N-(2-methoxyphenethyl)-4-(((S)-2-(m...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216181((R)-N-(2-methoxyphenethyl)-4-((diethylamino)methyl...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220382(4'-methyl-3-trifluoromethyl-biphenyl-4-carbonitril...)
Affinity DataIC50:  200nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220380(3'-hydroxy-3-trifluoromethyl-biphenyl-4-carbonitri...)
Affinity DataIC50:  229nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216204(CHEMBL394028 | N-(2-methoxyphenethyl)-4-(piperidin...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216206(CHEMBL393989 | N-(2-methoxyphenethyl)-4-(benzyloxy...)
Affinity DataIC50:  310nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220384(2',6'-dimethoxy-3-trifluoromethyl-biphenyl-4-carbo...)
Affinity DataIC50:  399nMAssay Description:Antagonist activity at human AR in MDA-MB453-MMTV-luci cells by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216191(CHEMBL232587 | N-(2,6-dichlorophenethyl)-4-((dieth...)
Affinity DataIC50:  430nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216187(CHEMBL232777 | N-(3-chlorophenethyl)-4-(benzyloxy)...)
Affinity DataIC50:  510nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216196(CHEMBL231776 | N-(2-methoxyphenethyl)-4-((diethyla...)
Affinity DataIC50:  540nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216183(CHEMBL233573 | N-(2-chlorophenethyl)-4-(benzyloxy)...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216207(CHEMBL233572 | N-(2-chlorophenethyl)-4-((diethylam...)
Affinity DataIC50:  840nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220382(4'-methyl-3-trifluoromethyl-biphenyl-4-carbonitril...)
Affinity DataIC50:  843nMAssay Description:Antagonist activity at human AR in MDA-MB453-MMTV-luci cells by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220388(3'-methoxy-3-trifluoromethyl-biphenyl-4-carbonitri...)
Affinity DataIC50:  955nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216208((S)-N-(2-methoxyphenethyl)-4-((diethylamino)methyl...)
Affinity DataIC50:  970nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220377(2',6'-dihydroxy-3-trifluoromethyl-biphenyl-4-carbo...)
Affinity DataIC50:  989nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220375(2'-methyl-3-trifluoromethyl-biphenyl-4-carbonitril...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human AR in MDA-MB453-MMTV-luci cells by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220381((4'-cyano-3'-trifluoromethyl-biphenyl-2-yloxy)-ace...)
Affinity DataIC50:  1.31E+3nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216186(CHEMBL232577 | N-(2-chlorophenethyl)-4-isopropoxy-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220387(2'-(2-hydroxy-ethoxy)-3-trifluoromethyl-biphenyl-4...)
Affinity DataIC50:  1.54E+3nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM25435(4-[(1S,2S)-2-hydroxycyclohexyl]-2-(trifluoromethyl...)
Affinity DataIC50:  1.60E+3nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-bound transcription factor site-1 protease(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50216203(4-diethylaminomethyl-N-pyrrolidin-3-yl-N-(2-o-toly...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human S1P expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220386(3'-methyl-3-trifluoromethyl-biphenyl-4-carbonitril...)
Affinity DataIC50:  1.90E+3nMAssay Description:Displacement of [3H]-DHT from human recombinant AR expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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