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Found 112 with Last Name = 'wakulchik' and Initial = 'm'
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137724((3aR,5S)-2-((S)-3-Methyl-2-{(S)-3-methyl-2-[(pyraz...)
Affinity DataKi:  17nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152750(2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carbonyl...)
Affinity DataKi:  20nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137721(2-(3-{[(1S,5S,6R)-2-((S)-3-Methyl-2-{(S)-3-methyl-...)
Affinity DataKi:  68nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152754(2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carbonyl...)
Affinity DataKi:  70nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137733((1S,5S,6R)-2-((S)-3,3-Dimethyl-2-{(S)-3-methyl-2-[...)
Affinity DataKi:  80nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152753((S)-2-((S)-3,3-Dimethyl-2-{(S)-3-methyl-2-[(pyrazi...)
Affinity DataKi:  80nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152748((S)-2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carb...)
Affinity DataKi:  80nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137713((S)-2-((S)-3-{[(1S,5S,6R)-4-Fluoro-2-((S)-3-methyl...)
Affinity DataKi:  82nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152751(2-((S)-2-{(S)-2-Cyclohexyl-2-[((R)-pyrazine-2-carb...)
Affinity DataKi:  90nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137718((1S,5S,6R)-2-((S)-3-Methyl-2-{(S)-3-methyl-2-[(pyr...)
Affinity DataKi:  90nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137720((1S,3aR,6aS)-2-((S)-3-Methyl-2-{(S)-3-methyl-2-[(p...)
Affinity DataKi:  123nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152755(2-((S)-2-{(S)-3-Methoxy-2-[(pyrazine-2-carbonyl)-a...)
Affinity DataKi:  150nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152752((S)-2-((S)-2-{(S)-3,3-Dimethyl-2-[(pyrazine-2-carb...)
Affinity DataKi:  160nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404057(CHEMBL118534)
Affinity DataKi:  170nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137722((S)-2-(3-{[(1S,5S,6R)-4,4-Difluoro-2-((S)-3-methyl...)
Affinity DataKi:  176nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152758((S)-2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carb...)
Affinity DataKi:  250nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137717((1S,5S,6R)-4-Fluoro-2-((S)-3-methyl-2-{(S)-3-methy...)
Affinity DataKi:  300nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137727((1S,5S,6R)-4-Fluoro-2-((S)-3-methyl-2-{(S)-3-methy...)
Affinity DataKi:  315nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137723((1S,5S)-4-Methoxymethoxy-2-((S)-3-methyl-2-{(S)-3-...)
Affinity DataKi:  332nMAssay Description:Cytotoxic activity against Protease in rat liver Huh-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137719((1S,5S,6R)-4,4-Difluoro-2-((S)-3-methyl-2-{(S)-3-m...)
Affinity DataKi:  370nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137725((1S,5S)-4-Methoxymethoxy-2-((S)-3-methyl-2-{(S)-3-...)
Affinity DataKi:  415nMAssay Description:Cytotoxic activity against Protease in rat liver Huh-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404055(CHEMBL118137)
Affinity DataKi:  500nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137728((5S,6R)-2-((S)-3-Methyl-2-{(S)-3-methyl-2-[(pyrazi...)
Affinity DataKi:  510nMAssay Description:Cytotoxic activity against Protease in rat liver Huh-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137714((1S,5S,6R)-2-((S)-3-Methyl-2-{(S)-3-methyl-2-[(pyr...)
Affinity DataKi:  625nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152756(2-((S)-3,3-Dimethyl-2-{(S)-2-phenyl-2-[(pyrazine-2...)
Affinity DataKi:  650nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152757((S)-2-((S)-2-{(S)-3-Cyclohexyl-2-[(pyrazine-2-carb...)
Affinity DataKi:  650nMAssay Description:Inhibition of HCV NS3 protease in the pNA based inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404062(CHEMBL325300)
Affinity DataKi:  710nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137716((1S,5S,6R)-2-((S)-3-Methyl-2-{(S)-3-methyl-2-[(pyr...)
Affinity DataKi:  880nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404063(CHEMBL118874)
Affinity DataKi:  940nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404058(CHEMBL120688)
Affinity DataKi:  1.36E+3nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137733((1S,5S,6R)-2-((S)-3,3-Dimethyl-2-{(S)-3-methyl-2-[...)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity towards human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137726((1S,5S,6R)-2-((S)-3-Methyl-2-{(S)-3-methyl-2-[(pyr...)
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50137715((1S,5S,6R)-2-((S)-3-Methyl-2-{(S)-3-methyl-2-[(pyr...)
Affinity DataKi:  2.60E+3nMAssay Description:Binding affinity towards Protease using PNA assay in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50133645(((S)-2-Methyl-1-{(1S,3aR,6aS)-1-[1-((S)-1-phenyl-e...)
Affinity DataKi:  3.00E+3nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152754(2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carbonyl...)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity towards human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152752((S)-2-((S)-2-{(S)-3,3-Dimethyl-2-[(pyrazine-2-carb...)
Affinity DataKi:  3.90E+3nMAssay Description:Binding affinity towards human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404059(CHEMBL120485)
Affinity DataKi:  4.60E+3nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50133641(((S)-2,2-Dimethyl-1-{(1S,3aR,6aS)-1-[1-((S)-1-phen...)
Affinity DataKi:  5.40E+3nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404061(CHEMBL264632)
Affinity DataKi:  5.50E+3nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404067(CHEMBL118965)
Affinity DataKi:  6.50E+3nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404065(CHEMBL118712)
Affinity DataKi:  6.50E+3nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152755(2-((S)-2-{(S)-3-Methoxy-2-[(pyrazine-2-carbonyl)-a...)
Affinity DataKi:  7.30E+3nMAssay Description:Binding affinity towards human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404060(CHEMBL120209)
Affinity DataKi:  7.40E+3nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404056(CHEMBL333595)
Affinity DataKi:  9.80E+3nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152753((S)-2-((S)-3,3-Dimethyl-2-{(S)-3-methyl-2-[(pyrazi...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity towards human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152748((S)-2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carb...)
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity towards human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152753((S)-2-((S)-3,3-Dimethyl-2-{(S)-3-methyl-2-[(pyrazi...)
Affinity DataKi:  1.50E+4nMAssay Description:Binding affinity towards human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404066(CHEMBL119565)
Affinity DataKi:  1.74E+4nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Human rhinovirus B)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50404064(CHEMBL120651)
Affinity DataKi:  2.91E+4nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50152750(2-((S)-2-{(S)-2-Cyclohexyl-2-[(pyrazine-2-carbonyl...)
Affinity DataKi:  4.00E+4nMAssay Description:Binding affinity towards human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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