Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:JAK1 (IC50): Recombinant human JAK1 catalytic domain (amino acids 850-1154; catalog number 08-144) is purchased from Carna Biosciences. 10 ng of JAK1...More data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:JAK1 (KI): For the determination of Ki, different amounts of compound are mixed with the enzyme and the enzymatic reaction is followed as a function ...More data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:JAK2 (Kd): JAK2 (Invitrogen, PV4210) is used at a final concentration of 5 nM. The binding experiment is performed in 50 mM Hepes pH 7.5, 0.01% Brij-...More data for this Ligand-Target Pair
Affinity DataIC50: 112nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 178nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:JAK2 (IC50): Recombinant human JAK2 catalytic domain (amino acids 808-1132; catalog number PV4210) is purchased from Invitrogen. 0.025 mU of JAK2 is ...More data for this Ligand-Target Pair
Affinity DataIC50: 186nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 209nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 219nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 257nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 355nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 372nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 417nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 417nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 427nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 427nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 427nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 437nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 562nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 562nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 562nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 676nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 776nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of human cathepsin S in human JY cells assessed as p10 accumulation by fluorescence-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 813nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.45E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.59E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.19E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.63E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.76E+3nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+4nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
Affinity DataKd: 0.100nMAssay Description:Binding affinity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKd: 0.900nMAssay Description:Binding affinity against HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKd: 0.400nMAssay Description:Binding affinity against HIV-1 proteaseMore data for this Ligand-Target Pair