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Found 23 with Last Name = 'wolfe' and Initial = 'mr'
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM75707((3R)-3-cyclopentyl-4-keto-3-phenyl-diazetidine-1,2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human MDA-MB-231 cells after 30 mins by fluorescence polarization activity-based protein profiling assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400986(CHEMBL1550905)
Affinity DataIC50:  600nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400986(CHEMBL1550905)
Affinity DataIC50:  600nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human HEK293T cells after 45 mins by fluorescence polarization activity-based protein profiling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400987(CHEMBL1316687)
Affinity DataIC50:  640nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydrolase RBBP9(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50314727(1-(thiazol-2-yl)ethanone O-cyclohexanecarbonyl oxi...)
Affinity DataIC50:  640nMAssay Description:Displacement of fluorophosphate-rhodamine from RBBP9 transfected in human HEK293T cells proteomes after 30 mins by SDS-PAGE gel fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydrolase RBBP9(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50314725(4-(cinnamoyloxyimino)-2,6-dimethylcyclohexa-2,5-di...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of fluorophosphate-rhodamine from RBBP9 transfected in human HEK293T cells proteomes after 30 mins by SDS-PAGE gel fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydrolase RBBP9(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50314728(4-(4-methoxybenzoyloxyimino)-2,6-dimethylcyclohexa...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of fluorophosphate-rhodamine from RBBP9 transfected in human HEK293T cells proteomes after 30 mins by SDS-PAGE gel fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydrolase RBBP9(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50314728(4-(4-methoxybenzoyloxyimino)-2,6-dimethylcyclohexa...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of fluorophosphate-rhodamine from recombinant RBBP9 transfected in mouse brain membrane proteomes after 30 mins by SDS-PAGE gel fluoresc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydrolase RBBP9(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50314729(1-(thiazol-2-yl)ethanone O-4-chlorobenzoyl oxime |...)
Affinity DataIC50:  1.90E+3nMAssay Description:Displacement of fluorophosphate-rhodamine from RBBP9 transfected in human HEK293T cells proteomes after 30 mins by SDS-PAGE gel fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400996(CHEMBL1699083)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400994(CHEMBL1719837)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400995(CHEMBL1706554)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400988(CHEMBL1701914)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400986(CHEMBL1550905)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in HEK293T cells after 1 hr by fluorescence polarization activity-based protein profiling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400993(CHEMBL1729870)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400989(CHEMBL1718102)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydrolase RBBP9(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50314726(1-(thiazol-2-yl)ethanone O-4-fluorobenzoyl oxime |...)
Affinity DataIC50:  5.70E+3nMAssay Description:Displacement of fluorophosphate-rhodamine from RBBP9 transfected in human HEK293T cells proteomes after 30 mins by SDS-PAGE gel fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400991(CHEMBL1711185)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydrolase RBBP9(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50216297(6',7',10,11-tetramethoxyemetan | CHEMBL50588 | Eme...)
Affinity DataIC50:  7.80E+3nMAssay Description:Displacement of fluorophosphate-rhodamine from RBBP9 transfected in human HEK293T cells proteomes after 30 mins by SDS-PAGE gel fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine hydrolase RBBP9(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50314724(1-(thiazol-2-yl)ethanone O-4-methoxybenzoyl oxime ...)
Affinity DataIC50:  9.20E+3nMAssay Description:Displacement of fluorophosphate-rhodamine from RBBP9 transfected in human HEK293T cells proteomes after 30 mins by SDS-PAGE gel fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400997(CHEMBL1521288)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human MDA-MB-231 cells after 30 mins by fluorescence polarization activity-based protein profiling assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400992(CHEMBL1701983)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400990(CHEMBL1723004)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed