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Found 207 with Last Name = 'zeng' and Initial = 'x'
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Hangzhou Medical College

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  30nMAssay Description:Binding affinity to wild type BCR-ABL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Hangzhou Medical College

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  30nMAssay Description:Binding affinity to FLT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Hangzhou Medical College

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  42nMAssay Description:Binding affinity to wild type BCR-ABL T315I mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  180nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of pNP-beta-GlcNAc as substrate by Lineweaver-burk ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  190nMAssay Description:Inhibition of human HexBMore data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507478(CHEMBL4440132)
Affinity DataKi:  600nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507463(CHEMBL4452208)
Affinity DataKi:  700nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507475(CHEMBL4435797)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507472(CHEMBL4548064)
Affinity DataKi:  900nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507470(CHEMBL4448965)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507462(CHEMBL4548738)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507464(CHEMBL4438655)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507475(CHEMBL4435797)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507463(CHEMBL4452208)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507472(CHEMBL4548064)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507469(CHEMBL4454357)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507470(CHEMBL4448965)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507469(CHEMBL4454357)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507461(CHEMBL4592668)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of human beta-N-acetylhexosaminidase using pNP-beta-GlcNAc as substrate by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507476(CHEMBL4555514)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507462(CHEMBL4548738)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507474(CHEMBL4455894)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50491601(CHEMBL2333316)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of human beta-N-acetylhexosaminidase using p-nitrophenyl glycoside as substrate by spectrometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507471(CHEMBL4540913)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507460(CHEMBL4471966)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using 4-Mu-GlcNAc as substrate measured after 30 mins by fluorescence as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507460(CHEMBL4471966)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate measured after 30 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507476(CHEMBL4555514)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507471(CHEMBL4540913)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507473(CHEMBL4559735)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507477(CHEMBL4564023)
Affinity DataKi:  8.30E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507468(CHEMBL4474777)
Affinity DataKi:  1.59E+4nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507464(CHEMBL4438655)
Affinity DataKi:  2.21E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507468(CHEMBL4474777)
Affinity DataKi:  2.47E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507460(CHEMBL4471966)
Affinity DataKi:  3.04E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate measured after 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507460(CHEMBL4471966)
Affinity DataKi:  3.04E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using 4-Mu-GlcNAc as substrate measured after 30 mins by fluorescence a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507473(CHEMBL4559735)
Affinity DataKi:  5.62E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507467(CHEMBL4544229)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human beta-N-acetylhexosaminidase using pNP-beta-GlcNAc as substrate by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50554249(CHEMBL4786058)
Affinity DataIC50:  0.160nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50554247(CHEMBL4778779)
Affinity DataIC50:  0.170nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50554244(CHEMBL4785851)
Affinity DataIC50:  0.170nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50554233(CHEMBL4755196)
Affinity DataIC50:  0.170nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50125052(CHEMBL3623004 | US10130617, Example 1 | US20240043...)
Affinity DataIC50:  0.180nMAssay Description:Induction of estrogen receptor degradation in human MCF7 cellsMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50125052(CHEMBL3623004 | US10130617, Example 1 | US20240043...)
Affinity DataIC50:  0.210nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hangzhou Medical College

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50554242(CHEMBL4742066)
Affinity DataIC50:  0.220nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50554235(CHEMBL4745817)
Affinity DataIC50:  0.240nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50554232(CHEMBL4791503)
Affinity DataIC50:  0.280nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Hangzhou Medical College

Curated by ChEMBL
LigandPNGBDBM50322535(3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N...)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of recombinant wild type Abl (unknown origin) in presence of [33P]-ATP by radiometric hotspot assayMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50554234(CHEMBL4763497)
Affinity DataIC50:  0.440nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Hangzhou Medical College

Curated by ChEMBL
LigandPNGBDBM50590371(CHEMBL5182618)
Affinity DataIC50:  0.540nMAssay Description:Binding affinity to human recombinant His-tagged full length ABL1 expressed in baculovirus expression system by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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