TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-9-cis-retinoic acid form human RXRalpha expressed in human Caco2 cells after 16 hrsMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]-9-cis-retinoic acid form human RXRalpha expressed in human Caco2 cells after 16 hrsMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Displacement of [3H]-9-cis-retinoic acid form human RXRalpha expressed in human Caco2 cells after 16 hrsMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataKi: 161nMAssay Description:Displacement of [3H]-9-cis-retinoic acid form human RXRalpha expressed in human Caco2 cells after 16 hrsMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: >8.00E+4nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 296nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 364nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 126nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 143nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 34nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 43nMAssay Description:Agonist activity at human recombinant Gal4-tagged RXRalpha expressed in human Caco2 cells assessed as receptor homodimerization after 24 hrs by mamma...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 420nMAssay Description:Agonist activity at human recombinant Gal4-tagged RXRalpha expressed in human Caco2 cells assessed as receptor homodimerization after 24 hrs by mamma...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Agonist activity at human recombinant Gal4-tagged RXRalpha expressed in human Caco2 cells assessed as receptor homodimerization after 24 hrs by mamma...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at human recombinant Gal4-tagged RXRalpha expressed in human Caco2 cells assessed as receptor homodimerization after 24 hrs by mamma...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University
Curated by ChEMBL
Arizona State University
Curated by ChEMBL
Affinity DataEC50: 1.82E+4nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair