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Found 171 with Last Name = 'de groote' and Initial = 'm'
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369514(CHEMBL605266)
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369512(CHEMBL605054)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067081(9-Fluoro-2-furan-2-yl-5,6-dihydro-[1,2,4]triazolo[...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50088475(1-(2-Methoxy-phenyl)-3-(2-pyridin-3-yl-quinazolin-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]DPCPX from rat cortical membranes Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  7.14nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50370152(CHEMBL610150)
Affinity DataKi:  7.20nMAssay Description:Binding affinity at human Adenosine A3 receptor expressed in HEK 293 cells by [125I]-AB MECA displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097451(4-Hydroxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369503(CHEMBL606312)
Affinity DataKi:  7.80nMAssay Description:Binding affinity athuman Adenosine A3 receptor expressed in HEK 293 cells by [125I]AB-MECA displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  9.47nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369509(CHEMBL605885)
Affinity DataKi:  9.70nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  11nMAssay Description:Binding affinity at human Adenosine A3 receptor expressed in HEK 293 cells by [125I]-AB MECA displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards rat Adenosine A1 receptor using [3H]-DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM35804((CGS21680) 3-(4-{2-[6-Amino-9-(5-ethylcarbamoylmet...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]NECA from Adenosine A2A receptor in rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  16nMAssay Description:Binding affinity at Adenosine A2A receptor in rat striatal membrane by [3H]ZM-241385 displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50067116(4-Methoxy-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benz...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101787(4-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067081(9-Fluoro-2-furan-2-yl-5,6-dihydro-[1,2,4]triazolo[...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101782(4-Nitro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097441(4-Methoxy-N-(2-phenyl-quinazolin-4-yl)-benzamide |...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097436(4-Methyl-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benza...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097440(CHEMBL165783 | N-(3-Phenyl-[1,2,4]thiadiazol-5-yl)...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369515(CHEMBL604636)
Affinity DataKi:  31nMAssay Description:Binding affinity athuman Adenosine A3 receptor expressed in HEK 293 cells by [125I]AB-MECA displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097432((Cis)-4-Methoxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097432((Cis)-4-Methoxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101783(4-Bromo-N-(4-phenyl-thiazol-2-yl)-benzamide | CHEM...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101781(4-Methyl-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101790(CHEMBL60334 | N-(4-Phenyl-thiazol-2-yl)-benzamide)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097442(4-Chloro-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benza...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50369511(CHEMBL605468)
Affinity DataKi:  41nMAssay Description:Binding affinity athuman Adenosine A3 receptor expressed in HEK 293 cells by [125I]AB-MECA displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097426((Cis)-4-Hydroxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097426((Cis)-4-Hydroxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101786(2,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101784(3,4-Dichloro-N-(4-phenyl-thiazol-2-yl)-benzamide |...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  63nMAssay Description:Ability to displace [3H]DPCPX from Adenosine A1 receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097431(4-Methoxy-N-(4-phenyl-thiazol-2-yl)-benzamide | 4-...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097431(4-Methoxy-N-(4-phenyl-thiazol-2-yl)-benzamide | 4-...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50088465(1-Phenyl-3-(3-pyridin-2-yl-isoquinolin-1-yl)-urea ...)
Affinity DataKi:  76nMAssay Description:Binding affinity of the compound was determined by its ability to displace [125I]-AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50101789(3-Chloro-N-(4-phenyl-thiazol-2-yl)-benzamide | CHE...)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097452(CHEMBL354004 | [4-(3-Phenyl-[1,2,4]thiadiazol-5-yl...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50067082((2-Amino-ethyl)-carbamic acid 4-(2,6-dioxo-1,3-dip...)
Affinity DataKi:  108nMAssay Description:Binding affinity of the compound was determined by its ability to displace [125I]-AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  110nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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