Report error Found 34 Enz. Inhib. hit(s) with Target = 'Inositol-trisphosphate 3-kinase A'
Affinity DataKi: 4.30E+3nM ΔG°: -31.9kJ/mole IC50: 1.02E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology
Curated by ChEMBL
Pohang University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:Binding affinity of the compound against recombinant plasmid rat brain IP3K by overexpressing in E. coliMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+4nMAssay Description:No assay is defined.More data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 1.82E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology
Curated by ChEMBL
Pohang University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2.74E+4nMAssay Description:Binding affinity of the compound against recombinant plasmid rat brain IP3K by overexpressing in E. coliMore data for this Ligand-Target Pair
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology
Curated by ChEMBL
Pohang University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2.78E+4nMAssay Description:Binding affinity of the compound against recombinant plasmid rat brain IP3K by overexpressing in E. coliMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 2.88E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology
Curated by ChEMBL
Pohang University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 3.94E+4nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 4.34E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology
Curated by ChEMBL
Pohang University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 4.37E+4nMAssay Description:Binding affinity of the compound against recombinant plasmid rat brain IP3K by overexpressing in E. coliMore data for this Ligand-Target Pair
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology
Curated by ChEMBL
Pohang University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 4.37E+4nMAssay Description:Binding affinity of the compound against recombinant plasmid rat brain IP3K by overexpressing in E. coliMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 5.71E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 6.76E+4nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology
Curated by ChEMBL
Pohang University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 9.00E+4nMAssay Description:Binding affinity of the compound against recombinant plasmid rat brain IP3K by overexpressing in E. coliMore data for this Ligand-Target Pair
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology
Curated by ChEMBL
Pohang University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against recombinant plasmid rat brain IP3K by overexpressing in E. coliMore data for this Ligand-Target Pair
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology
Curated by ChEMBL
Pohang University of Science & Technology
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity of the compound against recombinant plasmid rat brain IP3K by overexpressing in E. coliMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+5nMpH: 8.0 T: 37°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair