Report error Found 1701 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1'
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicles from SR3A cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicles from SR3A cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicles from SR3A cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Inhibition of MRP1 in human 2008/MRP1 cells by dixon plot analysisMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of MRP1 in human 2008/MRP1 cells by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicles from SR3A cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:TP_TRANSPORTER: inhibition of GSSG uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 380nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:TP_TRANSPORTER: inhibition of ATPase activity in Sf9 cells (membrane vesicles)More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibition of MRP1-mediated transport of [3H]LTC4 expressed in human HeLa T5 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:TP_TRANSPORTER: inhibition of GSSG uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Inhibition of human MRP1 expressed in Spodoptera frugiperda Sf9 cells assessed as inhibition of NEM-GS-induced vanadate-sensitive ATPase activity mea...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:TP_TRANSPORTER: inhibition of GSSG uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 950nMAssay Description:Inhibition of human MRP1 expressed in Spodoptera frugiperda Sf9 cells assessed as inhibition of NEM-GS-induced vanadate-sensitive ATPase activity mea...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 950nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in membrane vesicles from GLC4/ADR cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Noncompetitive inhibition of MRP1-mediated E2-17betaG transport in human MRP1 expressing HEK293 cells by Dixon plotMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of MRP1 transfected in human HeLa cells assessed as inhibition of [3H]LTC4 transport by rapid filtration assayMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of MRP1 transfected in human HeLa cells assessed as inhibition of [3H]LTC4 transport by rapid filtration assayMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of MRP1 transfected in human HeLa cells assessed as inhibition of [3H]LTC4 transport by rapid filtration assayMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of MRP1 transfected in human HeLa cells assessed as inhibition of [3H]LTC4 transport by rapid filtration assayMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of MRP1 transfected in human HeLa cells assessed as inhibition of [3H]LTC4 transport by rapid filtration assayMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (+3mM GSH) in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of MRP1 transfected in MDCK2 cells assessed as inhibition of calcein transportMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 8.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.32E+4nMAssay Description:Inhibition of MRP1 in human 2008/MRP1 cells by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.33E+4nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.34E+4nMAssay Description:Inhibition of MRP1 in human 2008/MRP1 cells by dixon plot analysisMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.08E+4nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (+3mM GSH) in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.70E+4nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.35E+5nMAssay Description:Inhibition of MRP1 in human 2008/MRP1 cells by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.40E+5nMAssay Description:Inhibition of MRP1 in human 2008/MRP1 cells by dixon plot analysisMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 0.765nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 0.960nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 1.16nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 1.25nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:TP_TRANSPORTER: cell accumulation in MCF7/MRP1-M6 cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:TP_TRANSPORTER: cell accumulation in MCF7/MRP1-M24 cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:TP_TRANSPORTER: cell accumulation in MCF7/MRP1-10 cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 6.32nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 6.96nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Human)
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
University of Texas M. D. Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 8.09nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
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