TargetNADP-dependent malic enzyme(Escherichia coli (strain K12))
Institute Of Chemical Physics
Curated by ChEMBL
Institute Of Chemical Physics
Curated by ChEMBL
Affinity DataKi: 5.70E+4nMAssay Description:Inhibition of Escherichia coli K-12 recombinant NAD-dependent malic enzyme by Dixon plotMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:In vitro inhibitory activity against human Carbonic anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory concentration against rat liver dihydrofolate reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory concentration against rat liver dihydrofolate reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:In vitro inhibitory activity against human Carbonic anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:In vitro inhibitory activity against human Carbonic anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:In vitro inhibitory concentration against rat liver dihydrofolate reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:In vitro inhibitory activity against human Carbonic anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:In vitro inhibitory activity against human Carbonic anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:In vitro inhibition of human Carbonic Anhydrase IIMore data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:In vitro inhibitory concentration against rat liver dihydrofolate reductase(DHFR)More data for this Ligand-Target Pair
Affinity DataIC50: 940nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of spermidine synthase activity was evaluatedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against Dihydrofolate reductase in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of spermidine synthase activity was evaluatedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+3nMAssay Description:50% inhibition of human carbonic anhydrase II assayed by CO2 hydration catalyzed by human erythrocytesMore data for this Ligand-Target Pair