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Found 13 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2'
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50241748(CHEMBL518059 | dihydro-beta-erythroidine)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50433569(CHEMBL2381563)
Affinity DataIC50:  6.00E+3nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50433566(CHEMBL2381566)
Affinity DataIC50:  1.78E+4nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50433572(CHEMBL2381568)
Affinity DataIC50:  5.23E+4nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50433573(CHEMBL2381570)
Affinity DataIC50:  4.80E+5nMAssay Description:Antagonist activity at (alpha4beta2)2alpha5 nAChR (unknown origin) expressed in Xenopus oocytes assessed as inhibition of acetylcholine-induced curre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50445610(CHEMBL3104068)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50445612(CHEMBL3103985)
Affinity DataEC50:  700nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50445609(CHEMBL3103999)
Affinity DataEC50:  1.30E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50445608(CHEMBL3104126)
Affinity DataEC50:  1.70E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50445607(CHEMBL3104079)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50445606(CHEMBL3103983)
Affinity DataEC50:  2.20E+3nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50445605(CHEMBL3104001)
Affinity DataEC50:  690nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/alpha-5/beta-2(Homo sapiens (Human))
University Of Chile

Curated by ChEMBL
LigandPNGBDBM50445611(CHEMBL3103988)
Affinity DataEC50:  790nMAssay Description:Positive allosteric modulation of human alpha4beta2alpha5 nACHR expressed in HEK-tsA201 cells assessed as potentiation of nicotine-induced current pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed