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Found 45 Enz. Inhib. hit(s) with Target = 'Tryptase delta'
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50475863(CHEMBL209054)
Affinity DataKi:  24nMAssay Description:Inhibition of mast cell tryptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50475860(CHEMBL424699)
Affinity DataKi:  34nMAssay Description:Inhibition of mast cell tryptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50475861(CHEMBL211733)
Affinity DataKi:  300nMAssay Description:Inhibition of mast cell tryptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50475865(CHEMBL212765)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of mast cell tryptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50475864(CHEMBL378085)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of mast cell tryptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50475862(CHEMBL379076)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of mast cell tryptaseMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217812(CHEMBL322526)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217627(CHEMBL110061)
Affinity DataIC50:  0.700nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217626(CHEMBL322538)
Affinity DataIC50:  0.700nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217622(CHEMBL443539)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217599(CHEMBL109888)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217801(CHEMBL111250)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217824(BMS-363130 | CHEMBL70738)
Affinity DataIC50: <1.70nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217823(CHEMBL111630)
Affinity DataIC50: <1.70nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217822(CHEMBL111173)
Affinity DataIC50: <1.70nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217818(CHEMBL440515)
Affinity DataIC50: <1.70nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217817(CHEMBL326209)
Affinity DataIC50: <1.70nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50120387((2S,3R)-3-((R)-1-Carbamimidoyl-piperidin-3-ylmethy...)
Affinity DataIC50: <1.70nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217819(CHEMBL109504)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217628(CHEMBL107493)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217624(CHEMBL321622)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50120368((2S,3R)-1-(4-tert-Butylcarbamoyl-piperazine-1-carb...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50120368((2S,3R)-1-(4-tert-Butylcarbamoyl-piperazine-1-carb...)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217813(CHEMBL302058)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217820(CHEMBL447534)
Affinity DataIC50:  4.60nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50220841(BMS-262084 | CHEMBL71037)
Affinity DataIC50:  5nMAssay Description:Inhibition of human lung tryptase using Z-glypro-arg-AMC incubated for 3 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217623(CHEMBL109947)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217805(CHEMBL111548)
Affinity DataIC50:  5.20nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217601(CHEMBL320744)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217601(CHEMBL320744)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217815(CHEMBL113591)
Affinity DataIC50:  6nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217625(CHEMBL326480)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217629(CHEMBL111270)
Affinity DataIC50:  9nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217816(CHEMBL432835)
Affinity DataIC50:  9nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217800(CHEMBL109254)
Affinity DataIC50:  9nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217811(CHEMBL109882)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217821(CHEMBL109733)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217600(CHEMBL109602)
Affinity DataIC50:  13nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217808(CHEMBL111141)
Affinity DataIC50:  18nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217814(CHEMBL324621)
Affinity DataIC50:  71nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217814(CHEMBL324621)
Affinity DataIC50:  71nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217598(CHEMBL320529)
Affinity DataIC50:  71nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217814(CHEMBL324621)
Affinity DataIC50:  204nMAssay Description:Inhibitory concentration against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM50217601(CHEMBL320744)
Affinity DataIC50:  5.38E+3nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM408717( N-[(3-fluoro-4-methoxypyridin-2-yl)methyl]-3-(met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human tryptase preincubated for 5 mins followed by substrate addition by fluorometer analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed