TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: >1.49E+3nMAssay Description:Inhibition of PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human PRKX using LRRASLG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human PRKX using LRRASLG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human PrkX by RFBA assayMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 326nMAssay Description:Inhibition of wild-type human partial length PRKX (M1 to F358 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of human wild type partial length PRKX (M1 to F358 residues) expressed in bacterial expression system by Kinomescan assayMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of PRKX (unknown origin)More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of human PrkX by RFBA assayMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PRKX (unknown origin)More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human full length PrKX using RRRLSFAEPG as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scin...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PRKX using [LRRASLG] as substrateMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant full length human GST-tagged PRKX expressed in baculovirus expression system using serine/threonine-1 peptide as substrate ...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 9.60E+5nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 1.30E+4nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 960nMAssay Description:Binding affinity to PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 42nMAssay Description:Binding affinity to PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 13nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 960nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 42nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 960nMAssay Description:Binding constant for full-length PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 13nMAssay Description:Binding constant for full-length PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PRKXMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 7.20nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 97nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: 5.80E+3nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit PRKX(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKX kinase domainMore data for this Ligand-Target Pair