Compile Data Set for Download or QSAR
maximum 50k data
Found 37 Enz. Inhib. hit(s) with all data for entry = 50012795
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560386(CHEMBL4743649)
Affinity DataIC50:  2nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212258(GS-4997 | Selonsertib)
Affinity DataIC50:  3nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50:  13nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50:  14nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560389(CHEMBL4744428)
Affinity DataIC50:  17nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560388(CHEMBL4753983)
Affinity DataIC50:  31nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212285(CHEMBL3891901)
Affinity DataIC50:  55nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50:  63nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50:  63nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50505941(CHEMBL4451125)
Affinity DataIC50:  100nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560387(CHEMBL4748155)
Affinity DataIC50:  130nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50:  200nMAssay Description:Inhibition of PRKKA1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50:  251nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50:  270nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50:  631nMAssay Description:Inhibition of MER (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of ROCK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of ITK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212282(CHEMBL3981026)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of p38 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of ROCK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of ITK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of ERBB4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of ERBB4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of EPHA3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of EPHA3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of p38 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of MER (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of HER4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of HER4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of PRKKA1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212258(GS-4997 | Selonsertib)
Affinity DataEC50:  2nMAssay Description:Inhibition of ASK1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560389(CHEMBL4744428)
Affinity DataEC50:  24nMAssay Description:Inhibition of ASK1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560389(CHEMBL4744428)
Affinity DataKd: <1nMAssay Description:Binding affinity to ASK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed