Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Tulahuen strain CYP51 expressed in Escherichia coli JM109More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of Trypanosoma cruzi CruzaineMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of Trypanosoma cruzi CruzaineMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of Trypanosoma cruzi CruzainMore data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of Trypanosoma cruzi CruzainMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of Trypanosoma cruzi CruzaineMore data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Inhibition of Trypanosoma cruzi CruzainMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of Trypanosoma cruzi CruzainMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Tulahuen strain CYP51 expressed in Escherichia coli JM109More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi Cruzain using Z-Phe-Arg-AMC as flurogenic substrateMore data for this Ligand-Target Pair
TargetTriosephosphate isomerase, glycosomal(Trypanosoma cruzi)
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Trypanosoma cruzi TIM expressed in Escherichia coli using glyceraldehyde 3-phosphate as substrate in presence of NADH/alphaGDPH measure...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Trypanosoma cruzi CruzainMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi CruzainMore data for this Ligand-Target Pair
TargetTriosephosphate isomerase, glycosomal(Trypanosoma cruzi)
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi TIMMore data for this Ligand-Target Pair
TargetTriosephosphate isomerase, glycosomal(Trypanosoma cruzi)
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi TIMMore data for this Ligand-Target Pair
TargetTriosephosphate isomerase, glycosomal(Trypanosoma cruzi)
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Trypanosoma cruzi TIMMore data for this Ligand-Target Pair
TargetTriosephosphate isomerase, glycosomal(Trypanosoma cruzi)
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi TIM using glyceraldehyde 3-phosphate as substrateMore data for this Ligand-Target Pair
TargetTriosephosphate isomerase, glycosomal(Trypanosoma cruzi)
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of Trypanosoma cruzi TIM expressed in Escherichia coli using glyceraldehyde 3-phosphate as substrate in presence of NADH/alphaGDPH measure...More data for this Ligand-Target Pair
TargetTriosephosphate isomerase, glycosomal(Trypanosoma cruzi)
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of Trypanosoma cruzi TIM expressed in Escherichia coli using glyceraldehyde 3-phosphate as substrate preincubated for 2 hrs in presence of...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi CruzaineMore data for this Ligand-Target Pair
TargetTriosephosphate isomerase, glycosomal(Trypanosoma cruzi)
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of Trypanosoma cruzi TIM expressed in Escherichia coli using glyceraldehyde 3-phosphate as substrate preincubated for 2 hrs in presence of...More data for this Ligand-Target Pair
TargetTriosephosphate isomerase, glycosomal(Trypanosoma cruzi)
Universidad De Navarra
Curated by ChEMBL
Universidad De Navarra
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi TIM using glyceraldehyde 3-phosphate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of Trypanosoma cruzi Cruzaine using Z-Phe-Arg-AMC as substrate preincubated for 15 mins measured for 10 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of Trypanosoma cruzi Tulahuen 2 Cruzain using Z-Phe-Arg-AMC as flurogenic substrate at 100 uM by spectrophotometry based analysis relative...More data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Inhibition of C-terminal His6-tagged Trypanosoma cruzi CYP51 expressed in Escherichia coli HMS174(DE3) assessed as dissociation constant by spectroph...More data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Displacement of [3H]-Eubricol from C-terminal His-tagged full-length Trypanosoma cruzi Tulahuen strain CYP51 expressed in Escherichia coli HMS174(DE3...More data for this Ligand-Target Pair