Affinity DataKi: 0.600nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Inhibition of cathepsin K (unknown origin) by fluorimetric assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase mutant (Tyr-181 to Cys)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase mutant (Tyr-181 to Cys)More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of cathepsin K (unknown origin) by fluorimetric assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase mutant (Tyr-181 to Leu)More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 840nMAssay Description:Inhibition of cathepsin K (unknown origin) by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
TargetMacrophage scavenger receptor types I and II(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of full-length MSR1 transfected in HEK293 cells by fluorimetryMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of HIV1 protease-mediated proteolysis of rabbit muscle lactate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV1 protease-mediated proteolysis of rabbit muscle lactate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human HMGCoA reductaseMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of HIV1 protease-mediated proteolysis of rabbit muscle lactate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIV1 protease-mediated proteolysis of rabbit muscle lactate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIV1 protease-mediated proteolysis of rabbit muscle lactate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of HIV1 protease-mediated proteolysis of rabbit muscle lactate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of cathepsin K (unknown origin) by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of cathepsin K (unknown origin) by fluorimetric assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetMacrophage scavenger receptor types I and II(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of full-length MSR1 transfected in HEK293 cells by fluorimetryMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against HIV-1 reverse transcriptase in scintillation proximity assayMore data for this Ligand-Target Pair