TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human IRR using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human IRR using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of IRR (unknown origin)More data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human INSRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of IRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant IRR (943 to 1266 residues) using myelin basic protein as substrate after 40 mins by [gamma-33ATP] by radiometric scin...More data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of INSRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human IRR using MBP as substrateMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human GST-tagged INSRR cytoplasmic domain expressed in baculovirus expression system using tyrosine-1 peptide as substrate ...More data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 1.82E+5nMAssay Description:Inhibition of human InsRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to INSRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 81nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 21nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 81nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 276nMAssay Description:Binding affinity to human IRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 430nMAssay Description:Binding affinity to INSRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRRMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 4.60E+3nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 600nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.60E+3nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair