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Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50133368'
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50133368(CHEMBL335950 | N-(2-(furan-2-yl)-8-(3-phenylpropyl...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H] DPCPX from human recombinant Adenosine A2B receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50133368(CHEMBL335950 | N-(2-(furan-2-yl)-8-(3-phenylpropyl...)
Affinity DataKi:  20nMAssay Description:Binding affinity to human adenosine A2b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50133368(CHEMBL335950 | N-(2-(furan-2-yl)-8-(3-phenylpropyl...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50133368(CHEMBL335950 | N-(2-(furan-2-yl)-8-(3-phenylpropyl...)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity against NECA stimulated cAMP accumulation in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50133368(CHEMBL335950 | N-(2-(furan-2-yl)-8-(3-phenylpropyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced adenylyl cyclase activityChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed