Found 4 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 2' and Ligand = 'BDBM50566697'
Affinity DataIC50: 40nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from 6His-Thr tagged BRD2 BD2/BD1 Y113A mutant (1 to 473 residues) (unknown origin) measured after 30...More data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+4nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from 6His-Thr tagged BRD2 BD1/BD2 Y386A mutant (1 to 473 residues) (unknown origin) measured after 30...More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding affinity to human partial length BRD2 BD 2 (E348 to D455 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.51E+4nMAssay Description:Binding affinity to human partial length BRD2 BD 1 expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair