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Found 6 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50061113'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50061113(3-(1',1'-dimethylheptyl)-6,6,9-trimethyl-6H-benzo[...)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50061113(3-(1',1'-dimethylheptyl)-6,6,9-trimethyl-6H-benzo[...)
Affinity DataKi:  1nMAssay Description:Binding affinity was determined for Cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50061113(3-(1',1'-dimethylheptyl)-6,6,9-trimethyl-6H-benzo[...)
Affinity DataKi:  2nMAssay Description:Compound was tested for inhibition of Adenylylcyclase in cannabinoid receptor 1 (CB1) .More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50061113(3-(1',1'-dimethylheptyl)-6,6,9-trimethyl-6H-benzo[...)
Affinity DataKi:  2nMAssay Description:Binding to Cannabinoid receptor 1 using African green monkey (COS-7) cells transfected with the cDNA of rat CB1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50061113(3-(1',1'-dimethylheptyl)-6,6,9-trimethyl-6H-benzo[...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity for Cannabinoid receptor 1 using African green monkey (COS-7) cells transfected with the cDNA of rat brain synaptosomal membrane pre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50061113(3-(1',1'-dimethylheptyl)-6,6,9-trimethyl-6H-benzo[...)
Affinity DataEC50:  0.180nMAssay Description:Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylylcyclase activity using African green monkey (COS-7) cells transfect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed