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Found 2 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor [668-1210,T790M,L858R]' and Ligand = 'BDBM50123163'
TargetEpidermal growth factor receptor [668-1210,T790M,L858R](Homo sapiens (Human))
Teligene

US Patent
LigandPNGBDBM50123163(CHEMBL3622672 | US9388160, 12)
Affinity DataIC50:  22nMpH: 7.4 T: 2°CAssay Description:The assay was performed using Kinase-Glo Plus luminescence kinase assay kit (Promega). The compounds were diluted in 10% DMSO and 5 μl of the dilu...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetEpidermal growth factor receptor [668-1210,T790M,L858R](Homo sapiens (Human))
Teligene

US Patent
LigandPNGBDBM50123163(CHEMBL3622672 | US9388160, 12)
Affinity DataIC50: <100nMpH: 7.4 T: 2°CAssay Description:The assay was performed using Kinase-Glo Plus luminescence kinase assay kit (Promega). The compounds were diluted in 10% DMSO and 5 μl of the dilu...More data for this Ligand-Target Pair
In DepthDetails US Patent