Found 2 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor [668-1210,T790M,L858R]' and Ligand = 'BDBM50123163'
TargetEpidermal growth factor receptor [668-1210,T790M,L858R](Homo sapiens (Human))
Teligene
US Patent
Teligene
US Patent
Affinity DataIC50: 22nMpH: 7.4 T: 2°CAssay Description:The assay was performed using Kinase-Glo Plus luminescence kinase assay kit (Promega). The compounds were diluted in 10% DMSO and 5 μl of the dilu...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor [668-1210,T790M,L858R](Homo sapiens (Human))
Teligene
US Patent
Teligene
US Patent
Affinity DataIC50: <100nMpH: 7.4 T: 2°CAssay Description:The assay was performed using Kinase-Glo Plus luminescence kinase assay kit (Promega). The compounds were diluted in 10% DMSO and 5 μl of the dilu...More data for this Ligand-Target Pair