Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'GABA A receptor alpha-1/beta-1/gamma-2' and Ligand = 'BDBM50503421'
TargetGABA A receptor alpha-1/beta-1/gamma-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50503421(CHEMBL4587325)
Affinity DataEC50:  1.48E+5nMAssay Description:Positive allosteric modulation of GABA-A alpha1beta1gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as increase in GAB...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGABA A receptor alpha-1/beta-1/gamma-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50503421(CHEMBL4587325)
Affinity DataEC50:  1.00E+4nMAssay Description:Positive allosteric modulation of GABA-A alpha1beta1(S290N)gamma2S mutant receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed