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Found 2 Enz. Inhib. hit(s) with Target = 'Glutaminase kidney isoform, mitochondrial [63-669]' and Ligand = 'BDBM416688'
TargetGlutaminase kidney isoform, mitochondrial [63-669](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM416688((2S)-2-ethoxy-2-[3-(3-methoxyazetidin-1-yl)phenyl]...)
Affinity DataIC50:  68.5nMAssay Description:A Glutamate Oxidase/AmplexRed coupled assay was used to measure the ability of compounds to bind to and inhibit the activity of GLS1 in vitro. 6His t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial [63-669](Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM416688((2S)-2-ethoxy-2-[3-(3-methoxyazetidin-1-yl)phenyl]...)
Affinity DataIC50:  131nMAssay Description:A Glutamate Oxidase/AmplexRed coupled assay was used to measure the ability of compounds to bind to and inhibit the activity of GLS1 in vitro. 6His t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent