Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50079575'
TargetHistamine H3 receptor(Homo sapiens (Human))
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataKi:  14nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Teva Global R & D.

Curated by ChEMBL
LigandPNGBDBM50079575(CHEMBL3417586)
Affinity DataEC50:  0.600nMAssay Description:Inverse agonist activity at human H3R expressed in CHO cells assessed as inhibition of RAMH-induced [35S]GTPgammaS binding relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed