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Found 2 Enz. Inhib. hit(s) with Target = 'Inhibitor of nuclear factor kappa-B kinase subunit beta' and Ligand = 'BDBM50244760'
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50244760((E)-4-{3-[3-Adamantan-1-yl-4-(2-methoxy-ethoxymeth...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of purified recombinant histidine-HA-tagged IKKbeta (unknown origin) expressed in SF9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50244760((E)-4-{3-[3-Adamantan-1-yl-4-(2-methoxy-ethoxymeth...)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of recombinant IKKbeta (unknown origin) using ulight-IkappaomegaBalpha as substrate after 2 hrs by LANCE ultra TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed