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Found 3 Enz. Inhib. hit(s) with Target = 'Integrin alpha-4/beta-1' and Ligand = 'BDBM50089005'
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech Chiroscience

Curated by ChEMBL
LigandPNGBDBM50089005((S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amin...)
Affinity DataIC50:  5nMAssay Description:Inhibition of CS-1 peptide binding to VLA-4 expressed in Ramos cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech Chiroscience

Curated by ChEMBL
LigandPNGBDBM50089005((S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amin...)
Affinity DataIC50:  34nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech Chiroscience

Curated by ChEMBL
LigandPNGBDBM50089005((S)-2-[((S)-3-Acetyl-thiazolidine-4-carbonyl)-amin...)
Affinity DataIC50:  410nMAssay Description:In vitro inhibition of binding of integrin alpha4-beta1 to immobilized VCAM-1 expressed on endothelial cell surface.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed