Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM209923'
TargetKappa-type opioid receptor(Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM209923(5'-Guanidinonaltrindole (5'-GNTI))
Affinity DataIC50:  0.0700nMAssay Description:For antagonist experiments, protein was preincubated with test compounds for 15 min prior to the addition of 100 nM U69,593 and [35S]GTPγS. Reac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
The Scripps Research Institute

LigandPNGBDBM209923(5'-Guanidinonaltrindole (5'-GNTI))
Affinity DataIC50:  0.800nMAssay Description:β-Arrestin2 translocation was also studied using the PathHunter® β-arrestin assay in CHO-K1 cells expressing the KOR (DiscoveRx, Fremont, C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed