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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50305819'
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50305819(1-(4-(thiophen-3-yl)benzyl)-5-(trifluoromethoxy)in...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M1 expressed in CHO cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50305819(1-(4-(thiophen-3-yl)benzyl)-5-(trifluoromethoxy)in...)
Affinity DataEC50:  1.19E+4nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay