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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50460765'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50460765(CHEMBL4229203)
Affinity DataEC50:  210nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M1 expressed in CHO cells assessed as potentiation of acetylcholine-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50460765(CHEMBL4229203)
Affinity DataEC50:  4.80E+3nMAssay Description:Allosteric agonist at human muscarinic acetylcholine receptor M1 expressed in CHO cells assessed as induction of calcium mobilization after 2.5 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed