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Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4' and Ligand = 'BDBM50264884'
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50264884(3-(2-chlorophenyl)-5-(5-methyl-1-(piperidin-4-yl)-...)
Affinity DataEC50:  18nMAssay Description:Activation of human alpha4beta2 nAChR assessed as potentiation of submaximal response to nicotine induced currentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Amgen

Curated by ChEMBL
LigandPNGBDBM50264884(3-(2-chlorophenyl)-5-(5-methyl-1-(piperidin-4-yl)-...)
Affinity DataEC50:  20nMAssay Description:Activation of rat alpha4beta2 nAChR by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed