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Found 4 Enz. Inhib. hit(s) with Target = 'Nucleotide-binding oligomerization domain-containing protein 2' and Ligand = 'BDBM50245040'
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50245040(CHEMBL4090558)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human NOD2 expressed in HEK-Blue cells assessed as induction of NF-kB transcriptional activity after 18 hrs by SEAP reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50245040(CHEMBL4090558)
Affinity DataEC50:  203nMAssay Description:Agonist activity at human human NOD2 expressed in HEK-Blue NOD2 reporter cells by colorimetry based SEAP assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50245040(CHEMBL4090558)
Affinity DataEC50:  99nMAssay Description:Agonist activity at NOD2 in HEK-Blue hNOD2 cells assessed as increase in NFkappaB activation incubated for 18 hrs by SEAP-based spectrophotometry ana...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Homo sapiens (Human))
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50245040(CHEMBL4090558)
Affinity DataEC50:  89nMAssay Description:Agonist activity at NOD2 in HEK-Blue hNOD2 cells assessed as increase in NFkappaB transactivation-mediated SEAP activity measured after 18 hrs by spe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed