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Found 2 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 3-kinase regulatory subunit alpha' and Ligand = 'BDBM318958'
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha(Homo sapiens (Human))
Teligene

US Patent
LigandPNGBDBM318958(N-(5-(2,6-dimorpholinopyrimidin-4-yl)-4-(trifluoro...)
Affinity DataIC50:  0.400nMAssay Description:An in vitro assay which determines the ability of a test compound to inhibit PI3K alpha activity: PI3 alpha (PIK3CA) kinase-tagged T7 phage strains w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha(Homo sapiens (Human))
Teligene

US Patent
LigandPNGBDBM318958(N-(5-(2,6-dimorpholinopyrimidin-4-yl)-4-(trifluoro...)
Affinity DataIC50:  32nMAssay Description:An in vitro assay which determines the ability of a test compound to inhibit PI3K alpha activity: PI3 delta (PIK3CD) kinase-tagged T7 phage strains w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent