Found 6 Enz. Inhib. hit(s) with Target = 'Proprotein convertase subtilisin/kexin type 9' and Ligand = 'BDBM217366' 
Affinity DataIC50: 1.40E+3nMAssay Description:For the peptide affinity determinations, biotinylated PCSK9 was immobilized to NeutrAvidin-coated MaxiSorp Immuno-Plates and incubated with a mixture...More data for this Ligand-Target Pair
Affinity DataEC50: 6.00E+3nMAssay Description:Inhibition of PCSK9 in human HepG2 cells assessed as increase in LDL uptakeMore data for this Ligand-Target Pair
Affinity DataKd: 700nMAssay Description:Binding affinity to human PCSK9More data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Inhibition of PCSK9 in human HepG2 cells assessed as restoration of LDLRMore data for this Ligand-Target Pair
Affinity DataKd: 700nMAssay Description:Binding affinity to recombinant human C-terminal His8-tagged PCSK9 expressed in Chinese hamster ovary cells by biolayer interferometryMore data for this Ligand-Target Pair
Affinity DataKd: 9.70E+3nMAssay Description:Binding affinity to human PCSK9 by surface plasmon resonanceMore data for this Ligand-Target Pair
