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Found 2 Enz. Inhib. hit(s) with Target = 'Pyruvate kinase PKLR' and Ligand = 'BDBM50028624'
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028624(CHEMBL3142978 | [6-(6-amino-9H-purin-9-yl)-2-methy...)
Affinity DataKi:  2.20E+6nMAssay Description:Inhibition of rat liver pyruvate kinase (PK-L) at 3.6 mMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyruvate kinase PKLR(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028624(CHEMBL3142978 | [6-(6-amino-9H-purin-9-yl)-2-methy...)
Affinity DataKi:  4.60E+6nMAssay Description:Inhibition of rat liver pyruvate kinase (PK-L); (relative inhibitory potency)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed