Found 5 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50109389'
Affinity DataKi: 30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain homogenates after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity of the compound for sigma-1 receptor by displacing [3H]-(+) pentazocineMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universita Degli Studi Di Bari
Curated by ChEMBL
Universita Degli Studi Di Bari
Curated by ChEMBL
Affinity DataKi: 309nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane without cerebellumMore data for this Ligand-Target Pair
Affinity DataKi: 309nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair