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Found 2 Enz. Inhib. hit(s) with Target = 'Sphingolipid delta(4)-desaturase DES1' and Ligand = 'BDBM523252'
TargetSphingolipid delta(4)-desaturase DES1(Homo sapiens (Human))TBA
LigandPNGBDBM523252((1r,4r)-4-(4- chlorophenyl)- N-(5-hydroxy- pyridin...)
Affinity DataIC50:  1nMAssay Description:Negative log concentration of antagonist was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSphingolipid delta(4)-desaturase DES1(Homo sapiens (Human))TBA
LigandPNGBDBM523252((1r,4r)-4-(4- chlorophenyl)- N-(5-hydroxy- pyridin...)
Affinity DataIC50:  1nMAssay Description:Jurkat clone E6-1 cells were grown and then seeded at 106 cells/mL in a 96-well plate (400 μL in each well. The cells were administered 100 _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent