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Found 4 Enz. Inhib. hit(s) with Target = 'Toll-like receptor 1' and Ligand = 'BDBM50511993'
TargetToll-like receptor 1(Homo sapiens)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50511993(CHEMBL4472879)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at TLR1/2 in human THP-1 cells assessed as increase in TNF-alpha release incubated for 4 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 1(Homo sapiens)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50511993(CHEMBL4472879)
Affinity DataEC50:  1.30nMAssay Description:In vitro histamine H3 receptor antagonist activity was determined on guinea pig jejunumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetToll-like receptor 1(Homo sapiens)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50511993(CHEMBL4472879)
Affinity DataEC50:  0.110nMAssay Description:Histamine H2-receptor activity on isolated spontaneously beating guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetToll-like receptor 1(Homo sapiens)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50511993(CHEMBL4472879)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at TLR1/TLR2 in human THP-1 derived macrophages assessed as stimulation of TNF alpha release measured for 4 hrs by ELISA based assayMore data for this Ligand-Target Pair
In DepthDetails PubMed