Affinity DataEC50: 0.110nMAssay Description:Agonist activity at TLR1/2 in human THP-1 cells assessed as increase in TNF-alpha release incubated for 4 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:In vitro histamine H3 receptor antagonist activity was determined on guinea pig jejunumMore data for this Ligand-Target Pair
Affinity DataEC50: 0.110nMAssay Description:Histamine H2-receptor activity on isolated spontaneously beating guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataEC50: 0.110nMAssay Description:Agonist activity at TLR1/TLR2 in human THP-1 derived macrophages assessed as stimulation of TNF alpha release measured for 4 hrs by ELISA based assayMore data for this Ligand-Target Pair