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TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50247011(CHEMBL4080419)
Affinity DataKi:  0.0110nMAssay Description:Competitive inhibition of recombinant human BChE using butyrylthiocholine iodide as substrate at pH 8 by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2019
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50247011(CHEMBL4080419)
Affinity DataKi:  0.0110nMAssay Description:Competitive inhibition of recombinant human BChE using butyrylthiocholine iodide as substrate at pH 8 by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2019
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50005193(CHEMBL3099496)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of human butyrylcholine esteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50599186(CHEMBL5201089)
Affinity DataKi:  0.0940nMAssay Description:Inhibition of human BChE assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50234795(CHEMBL4089082)
Affinity DataKi:  0.131nMAssay Description:Inhibition of human serum BChE using butyrylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2019
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8963(N-[7-(1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-...)
Affinity DataKi:  0.163nMAssay Description:Competitive inhibition of recombinant human BChE using butyrylthiocholine iodide as substrate at pH 8 by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2019
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50604405(CHEMBL5186889)
Affinity DataKi:  0.180nMAssay Description:Binding affinity to human recombinant BChE in enzyme-inhibitor complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50604405(CHEMBL5186889)
Affinity DataKi:  0.180nMAssay Description:Binding affinity to human recombinant BChE in enzyme-substrate-inhibitor complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271323(N-{4-[(1,2,3, 4-Tetrahydroacridin-9-yl)amino]butyl...)
Affinity DataKi:  0.270nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8971(CHEMBL129108 | N-[8-(1,2,3,4-tetrahydroacridin-9-y...)
Affinity DataKi:  0.400nMAssay Description:Inhibition of Equine ButyrylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271468(N-Ethyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(...)
Affinity DataKi:  0.435nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50599167(CHEMBL5195228)
Affinity DataKi:  0.610nMAssay Description:Inhibition of human BChE assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271325(N-{4-[(1,2,3,4-Tetrahydroacridin-9-yl)amino]butyl}...)
Affinity DataKi:  0.725nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8977(N-[3-(1,2,3,4-Tetrahydroacridin-9-ylamino)propyl]-...)
Affinity DataKi:  0.740nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271324(N-(1,2,3,4-Tetrahydroacridin-9-yl)-N-(3-(1,2,3,4-t...)
Affinity DataKi:  0.779nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271367(N-Methyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[...)
Affinity DataKi:  0.819nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271367(N-Methyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[...)
Affinity DataKi:  0.820nMAssay Description:Inhibition of human butyrylcholine esteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271472(1,3-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]eth...)
Affinity DataKi:  0.924nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468733(CHEMBL4294570)
Affinity DataKi:  1.10nMAssay Description:Competitive inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50620155(CHEMBL5435281)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human BChE assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271470(N-(2-Hydroxyethyl)-N-(1,2,3,4-tetrahydroacridin-9-...)
Affinity DataKi:  1.19nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50265253((S)-2-amino-3-(1H-indol-3-yl)-N-(2-(1,2,3,4-tetrah...)
Affinity DataKi:  1.33nMAssay Description:Inhibition of human recombinant BChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8971(CHEMBL129108 | N-[8-(1,2,3,4-tetrahydroacridin-9-y...)
Affinity DataKi:  1.65nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8971(CHEMBL129108 | N-[8-(1,2,3,4-tetrahydroacridin-9-y...)
Affinity DataKi:  1.65nMAssay Description:Inhibition of human recombinant BChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8971(CHEMBL129108 | N-[8-(1,2,3,4-tetrahydroacridin-9-y...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human butyrylcholine esteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468736(CHEMBL4283585)
Affinity DataKi:  1.70nMAssay Description:Competitive inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50265256((S)-1-(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethy...)
Affinity DataKi:  1.77nMAssay Description:Inhibition of human recombinant BChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271473(2,6-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]eth...)
Affinity DataKi:  1.87nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50265252((S)-tert-butyl 3-(1H-indol-3-yl)-1-oxo-1-(2-(1,2,3...)
Affinity DataKi:  1.87nMAssay Description:Inhibition of human recombinant BChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8969(CHEMBL131410 | N,N-bis[3-(1,2,3,4-tetrahydroacridi...)
Affinity DataKi:  2nMAssay Description:Inhibition of Equine ButyrylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8963(N-[7-(1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-...)
Affinity DataKi:  2nMAssay Description:Inhibition of Equine ButyrylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50027375(CHEMBL3338394)
Affinity DataKi:  2.70nMAssay Description:Inhibition of recombinant human BChE at 50 nM by stopped flow apparatus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50604404(CHEMBL5186857)
Affinity DataKi:  3nMAssay Description:Binding affinity to human recombinant BChE in enzyme-inhibitor complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8975(CHEMBL179192 | N-[3-(1,2,3,4-Tetrahydroacridin-9-y...)
Affinity DataKi:  3.13nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271471(1,4-bis[3-(1,2,3,4-Tetrahydroacridin-9-yl)aminopro...)
Affinity DataKi:  3.22nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50219206(Anthracen-9-yl (10H-phenothiazine-10yl) methanone,...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of human plasma BuChE activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50626851(CHEMBL5402537)
Affinity DataKi:  4nMAssay Description:Competitive inhibition of human BuChE using butyrylthiocholine iodide as substrate assessed as inhibition constant preincubated with enzyme for 5 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271469(N-Allyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(...)
Affinity DataKi:  4.19nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271518(1,3-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]eth...)
Affinity DataKi:  5.04nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8965(CHEMBL338755 | methylbis[3-(1,2,3,4-tetrahydroacri...)
Affinity DataKi:  6nMAssay Description:Inhibition of Equine ButyrylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50604404(CHEMBL5186857)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to human recombinant BChE in enzyme-substrate-inhibitor complexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant BChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataKi:  7nMAssay Description:Inhibition of Equine ButyrylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataKi:  7nM ΔG°:  -11.1kcal/molepH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by E llman. Inhibition of enzyme activity was measured over a substrate c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50271519(3,4-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]eth...)
Affinity DataKi:  7.29nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50056112(CHEMBL3326702)
Affinity DataKi:  8.10nMAssay Description:Inhibition of human BChE assessed as acetylthiocholine hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50005192(CHEMBL3099497)
Affinity DataKi:  8.30nMAssay Description:Inhibition of human butyrylcholine esteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50555837(CHEMBL4747577)
Affinity DataKi:  8.30nMAssay Description:Mixed inhibition of human butyrylcholinesterase assessed as affinity towards free enzyme using butyrylthiocholine iodide as substrate measured by Ell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8976(N-Methyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-[4-(...)
Affinity DataKi:  8.59nMAssay Description:Inhibition of human recombinant BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
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