Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nM ΔG°: -53.3kJ/molepH: 7.4 T: 2°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
Affinity DataKi: 0.770nMAssay Description:Binding affinity at Vasopressin V2 receptor, performed using [3H]-AVP on rat kidneyMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]AVP from V2 receptor in Wistar rat kidney membranes incubated for 60 mins by microplate scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataKi: 12.7nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 19nM ΔG°: -43.8kJ/molepH: 7.4 T: 2°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Inhibition of [3H]-arginine vasopressin binding to rat kidney medulla Vasopressin V2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Inhibition of [3H]-arginine vasopressin binding to rat kidney medulla Vasopressin V2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Binding affinity against Vasopressin receptor in rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity against Vasopressin receptor in rat kidney medullaMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Binding affinity against Vasopressin receptor in rat kidney medullaMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity against Vasopressin receptor in rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Binding affinity towards rat kidney Vasopressin V2 receptor by using functional assayMore data for this Ligand-Target Pair
Affinity DataKi: 168nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]-vasopressin from vasopressin V2 receptor in rat kidney tissueMore data for this Ligand-Target Pair