Compile Data Set for Download or QSAR
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Found 38 Enz. Inhib. hit(s) with all data for entry = 50014863
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148441(2-{4-[2-(1,2,3,4-Tetrahydro-quinolin-7-yloxy)-etho...)
Affinity DataEC50:  140nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50064455(4-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-be...)
Affinity DataEC50:  83nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148440(2-{4-[2-(5,6,7,8-Tetrahydro-naphthalen-2-yloxy)-et...)
Affinity DataEC50:  4.68E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  2.88E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  1.46E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148444(2-{4-[2-(Naphthalen-2-yloxy)-ethoxy]-benzyl}-malon...)
Affinity DataEC50:  1.12E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148443(2-{4-[2-(1,2,3,4-Tetrahydro-quinolin-7-yloxy)-etho...)
Affinity DataEC50:  3.80E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148445(2-{4-[2-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-na...)
Affinity DataEC50:  150nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148446(2-{4-[2-(1,2,3,4-Tetrahydro-quinolin-7-yloxy)-etho...)
Affinity DataEC50:  170nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148447(2-{4-[2-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-na...)
Affinity DataEC50:  830nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148448(2-{4-[2-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-na...)
Affinity DataEC50:  2.05E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148449(2-{4-[2-(Naphthalen-2-yloxy)-ethoxy]-benzyl}-malon...)
Affinity DataEC50:  250nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148444(2-{4-[2-(Naphthalen-2-yloxy)-ethoxy]-benzyl}-malon...)
Affinity DataEC50:  44nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148450(2-{4-[2-(Naphthalen-2-yloxy)-ethoxy]-benzyl}-malon...)
Affinity DataEC50:  530nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148441(2-{4-[2-(1,2,3,4-Tetrahydro-quinolin-7-yloxy)-etho...)
Affinity DataEC50:  2.88E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148443(2-{4-[2-(1,2,3,4-Tetrahydro-quinolin-7-yloxy)-etho...)
Affinity DataEC50:  90nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148450(2-{4-[2-(Naphthalen-2-yloxy)-ethoxy]-benzyl}-malon...)
Affinity DataEC50:  70nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148451(2-{4-[2-(5,6,7,8-Tetrahydro-naphthalen-2-yloxy)-et...)
Affinity DataEC50:  3.31E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  3.62E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148450(2-{4-[2-(Naphthalen-2-yloxy)-ethoxy]-benzyl}-malon...)
Affinity DataEC50:  1.27E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148451(2-{4-[2-(5,6,7,8-Tetrahydro-naphthalen-2-yloxy)-et...)
Affinity DataEC50:  1.50E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148444(2-{4-[2-(Naphthalen-2-yloxy)-ethoxy]-benzyl}-malon...)
Affinity DataEC50:  1.05E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148452(2-{4-[2-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-na...)
Affinity DataEC50:  90nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148440(2-{4-[2-(5,6,7,8-Tetrahydro-naphthalen-2-yloxy)-et...)
Affinity DataEC50:  2.11E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  140nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148442(2-{4-[2-(5,6,7,8-Tetrahydro-naphthalen-2-yloxy)-et...)
Affinity DataEC50:  2.45E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148453(2-{4-[2-(5,6,7,8-Tetrahydro-naphthalen-2-yloxy)-et...)
Affinity DataEC50:  3.43E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148446(2-{4-[2-(1,2,3,4-Tetrahydro-quinolin-7-yloxy)-etho...)
Affinity DataEC50:  3.16E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148443(2-{4-[2-(1,2,3,4-Tetrahydro-quinolin-7-yloxy)-etho...)
Affinity DataEC50:  3.09E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148446(2-{4-[2-(1,2,3,4-Tetrahydro-quinolin-7-yloxy)-etho...)
Affinity DataEC50:  3.16E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148454(2-Bromo-hexadecanoic acid | CHEMBL118417)
Affinity DataEC50:  3.72E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148441(2-{4-[2-(1,2,3,4-Tetrahydro-quinolin-7-yloxy)-etho...)
Affinity DataEC50:  3.62E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148451(2-{4-[2-(5,6,7,8-Tetrahydro-naphthalen-2-yloxy)-et...)
Affinity DataEC50:  30nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148449(2-{4-[2-(Naphthalen-2-yloxy)-ethoxy]-benzyl}-malon...)
Affinity DataEC50:  2.63E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-delta (PPAR delta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148449(2-{4-[2-(Naphthalen-2-yloxy)-ethoxy]-benzyl}-malon...)
Affinity DataEC50:  3.02E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  1.55E+4nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50064455(4-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-be...)
Affinity DataEC50:  1.90E+3nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-alpha (PPAR alpha)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Research Institute Of Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50148442(2-{4-[2-(5,6,7,8-Tetrahydro-naphthalen-2-yloxy)-et...)
Affinity DataEC50:  690nMAssay Description:In vitro transcription activation on human peroxisome proliferator activated receptor-gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed