Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50037478
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118812BDBM50118812(CHEMBL119709 | (3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-io...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370531BDBM50370531(CHEMBL608755)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370529BDBM50370529(CHEMBL611091)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370535BDBM50370535(CHEMBL611095)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370539BDBM50370539(CHEMBL611104)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370536BDBM50370536(CHEMBL610845)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21220BDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKi:  12.2nMAssay Description:Displacement of [3H]CGS-21680 binding to Adenosine A2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370543BDBM50370543(CHEMBL610849)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370537BDBM50370537(CHEMBL610814)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21220BDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKi:  18.2nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370528BDBM50370528(CHEMBL610846)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370542BDBM50370542(CHEMBL610589)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370534BDBM50370534(CHEMBL611089)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370541BDBM50370541(CHEMBL610847)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370527BDBM50370527(CHEMBL611090)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370524BDBM50370524(CHEMBL610837)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370525BDBM50370525(CHEMBL610584)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370532BDBM50370532(CHEMBL610830)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370538BDBM50370538(CHEMBL610579)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370526BDBM50370526(CHEMBL611092)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370533BDBM50370533(CHEMBL611099)
Affinity DataKi:  25nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21220BDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKi:  34.8nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370540BDBM50370540(CHEMBL610829)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370535BDBM50370535(CHEMBL611095)
Affinity DataIC50: 42nMAssay Description:Inhibition of (10 uM) forskolin-mediated cAMP production in CHO cells expressing human Adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370529BDBM50370529(CHEMBL611091)
Affinity DataIC50: 50nMAssay Description:Inhibition of (10 uM) forskolin-mediated cAMP production in CHO cells expressing human Adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118812BDBM50118812(CHEMBL119709 | (3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-io...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370531BDBM50370531(CHEMBL608755)
Affinity DataIC50: 55nMAssay Description:Inhibition of (10 uM) forskolin-mediated cAMP production in CHO cells expressing human Adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118812BDBM50118812(CHEMBL119709 | (3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-io...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]CGS-21680 binding to Adenosine A2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370539BDBM50370539(CHEMBL611104)
Affinity DataIC50: 65nMAssay Description:Inhibition of (10 uM) forskolin-mediated cAMP production in CHO cells expressing human Adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370530BDBM50370530(CHEMBL610580)
Affinity DataKi:  80nMAssay Description:Displacement of [125I]AB-MECA binding to Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370535BDBM50370535(CHEMBL611095)
Affinity DataKi:  206nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370540BDBM50370540(CHEMBL610829)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370524BDBM50370524(CHEMBL610837)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370528BDBM50370528(CHEMBL610846)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370542BDBM50370542(CHEMBL610589)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370536BDBM50370536(CHEMBL610845)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370527BDBM50370527(CHEMBL611090)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370533BDBM50370533(CHEMBL611099)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370526BDBM50370526(CHEMBL611092)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370531BDBM50370531(CHEMBL608755)
Affinity DataKi:  325nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370543BDBM50370543(CHEMBL610849)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370525BDBM50370525(CHEMBL610584)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370529BDBM50370529(CHEMBL611091)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370539BDBM50370539(CHEMBL611104)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370538BDBM50370538(CHEMBL610579)
Affinity DataKi:  415nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370530BDBM50370530(CHEMBL610580)
Affinity DataKi:  445nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370541BDBM50370541(CHEMBL610847)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370534BDBM50370534(CHEMBL611089)
Affinity DataKi:  725nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370532BDBM50370532(CHEMBL610830)
Affinity DataKi:  730nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370537BDBM50370537(CHEMBL610814)
Affinity DataKi:  750nMAssay Description:Displacement of [3H]CHA binding to Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
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