Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50017399
Affinity DataEC50: 2.40nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 20.2nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 21.5nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 32.5nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 38.5nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 41nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 54nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 56nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 61nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 64nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 68nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 71nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 72nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 77nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 83nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 87nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 89nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 98nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 102nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 106nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 107nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 116nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 119nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 123nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 131nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 137nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 141nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 168nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 192nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 194nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 203nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 207nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 209nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 221nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 221nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 284nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 296nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 309nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 333nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Mouse)
University of California San Francisco
Curated by ChEMBL
University of California San Francisco
Curated by ChEMBL
Affinity DataEC50: 371nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 800nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair




























