Compile Data Set for Download or QSAR
maximum 50k data
Found 84 Enz. Inhib. hit(s) with all data for entry = 4669
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81643(4,5-Dihydro-(1H)-pyrazole derivative, 1k)
Affinity DataIC50:  8.60nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81639(4,5-Dihydro-(1H)-pyrazole derivative, 1g)
Affinity DataIC50:  8.80nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50164871(1-(3,5-Diphenyl-4,5-dihydro-pyrazol-1-yl)-ethanone...)
Affinity DataIC50:  9nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81642(4,5-Dihydro-(1H)-pyrazole derivative, 1j)
Affinity DataIC50:  10nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81659(4,5-Dihydro-(1H)-pyrazole derivative, 3c)
Affinity DataIC50:  10nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297427(1-(5-(3,4-dimethoxyphenyl)-3-phenyl-4,5-dihydro-1H...)
Affinity DataIC50:  10nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81638(4,5-Dihydro-(1H)-pyrazole derivative, 1e)
Affinity DataIC50:  10nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81660(4,5-Dihydro-(1H)-pyrazole derivative, 3d)
Affinity DataIC50:  10nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81652(4,5-Dihydro-(1H)-pyrazole derivative, 2i)
Affinity DataIC50:  14nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297422(1-(3-(2,6-dihydroxyphenyl)-5-m-tolyl-4,5-dihydro-1...)
Affinity DataIC50:  28nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81666(4,5-Dihydro-(1H)-pyrazole derivative, 3l)
Affinity DataIC50:  50nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297422(1-(3-(2,6-dihydroxyphenyl)-5-m-tolyl-4,5-dihydro-1...)
Affinity DataIC50:  60nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81651(4,5-Dihydro-(1H)-pyrazole derivative, 2g)
Affinity DataIC50:  72nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297423(4,5-Dihydro-(1H)-pyrazole derivative, 2h | 4-(1-ph...)
Affinity DataIC50:  73nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81654(4,5-Dihydro-(1H)-pyrazole derivative, 2k)
Affinity DataIC50:  86nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81645(4,5-Dihydro-(1H)-pyrazole derivative, 1n)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81644(4,5-Dihydro-(1H)-pyrazole derivative, 1l)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81641(4,5-Dihydro-(1H)-pyrazole derivative, 1i)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297429(1-(3-phenyl-5-o-tolyl-4,5-dihydro-1H-pyrazol-1-yl)...)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297428(1-(3-(2,4-dihydroxyphenyl)-5-phenyl-4,5-dihydro-1H...)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81638(4,5-Dihydro-(1H)-pyrazole derivative, 1e)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81669(4,5-Dihydro-(1H)-pyrazole derivative, 3o)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81668(4,5-Dihydro-(1H)-pyrazole derivative, 3n)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81667(4,5-Dihydro-(1H)-pyrazole derivative, 3m)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297433(1-(3-(3,4-dimethoxyphenyl)-4,5-dihydro-1H-pyrazol-...)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81658(4,5-Dihydro-(1H)-pyrazole derivative, 3b)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81657(4,5-Dihydro-(1H)-pyrazole derivative, 3a)
Affinity DataIC50:  100nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81653(4,5-Dihydro-(1H)-pyrazole derivative, 2j)
Affinity DataIC50:  110nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297435(1-(3-(2,5-dimethoxyphenyl)-4,5-dihydro-1H-pyrazol-...)
Affinity DataIC50:  200nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81661(4,5-Dihydro-(1H)-pyrazole derivative, 3e)
Affinity DataIC50:  200nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81664(4,5-Dihydro-(1H)-pyrazole derivative, 3h)
Affinity DataIC50:  230nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81662(4,5-Dihydro-(1H)-pyrazole derivative, 3f)
Affinity DataIC50:  240nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81663(4,5-Dihydro-(1H)-pyrazole derivative, 3g)
Affinity DataIC50:  290nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81665(4,5-Dihydro-(1H)-pyrazole derivative, 3k)
Affinity DataIC50:  300nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81637(4,5-Dihydro-(1H)-pyrazole derivative, 1c)
Affinity DataIC50:  1.00E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81652(4,5-Dihydro-(1H)-pyrazole derivative, 2i)
Affinity DataIC50:  1.00E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81654(4,5-Dihydro-(1H)-pyrazole derivative, 2k)
Affinity DataIC50:  1.45E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81655(4,5-Dihydro-(1H)-pyrazole derivative, 2l)
Affinity DataIC50:  1.80E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81640(4,5-Dihydro-(1H)-pyrazole derivative, 1h)
Affinity DataIC50:  2.00E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297423(4,5-Dihydro-(1H)-pyrazole derivative, 2h | 4-(1-ph...)
Affinity DataIC50:  3.00E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81656(4,5-Dihydro-(1H)-pyrazole derivative, 2m)
Affinity DataIC50:  3.00E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM50297431(1-phenyl-3-p-tolyl-4,5-dihydro-1H-pyrazole | 4,5-D...)
Affinity DataIC50:  6.90E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81649(4,5-Dihydro-(1H)-pyrazole derivative, 2d)
Affinity DataIC50:  7.40E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81646(4,5-Dihydro-(1H)-pyrazole derivative, 2a)
Affinity DataIC50:  9.80E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81648(4,5-Dihydro-(1H)-pyrazole derivative, 2c)
Affinity DataIC50:  9.90E+3nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81647(4,5-Dihydro-(1H)-pyrazole derivative, 2b)
Affinity DataIC50:  1.00E+4nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81653(4,5-Dihydro-(1H)-pyrazole derivative, 2j)
Affinity DataIC50:  1.25E+4nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81656(4,5-Dihydro-(1H)-pyrazole derivative, 2m)
Affinity DataIC50:  1.70E+4nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81669(4,5-Dihydro-(1H)-pyrazole derivative, 3o)
Affinity DataIC50:  1.90E+4nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
UniversitÀ

LigandPNGBDBM81658(4,5-Dihydro-(1H)-pyrazole derivative, 3b)
Affinity DataIC50:  2.00E+4nMAssay Description:Monoamine oxidase inhibitory activity of derivatives of 4, dihydro-(1H)-pyrazole.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 84 total ) | Next | Last >>
Jump to: