Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50038312
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 0.00800nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0630nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0780nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0970nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 64nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 390nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 550nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 770nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.46E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.75E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.05E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair





