Compile Data Set for Download or QSAR
maximum 50k data
Found 68 Enz. Inhib. hit(s) with all data for entry = 50026921
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244455((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3,5-dichl...)
Affinity DataIC50:  3.90nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245098((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(3,5-dichloroph...)
Affinity DataIC50:  4nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245102((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3-methane...)
Affinity DataIC50:  5nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245060((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(4-trifluoromet...)
Affinity DataIC50:  6nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245099((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(2,2,4,4-t...)
Affinity DataIC50:  6nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244507((R)-3-{4-[3-(3-Bromo-5-trifluoromethylphenyl)-1-(4...)
Affinity DataIC50:  7nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244506((R)-3-{4-[3-(3-Bromophenyl)-1-(4-cyclohexylphenyl)...)
Affinity DataIC50:  8nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244457((R)-trans-3-{4-[3-(3,5-Bis(trifluoromethyl)phenyl)...)
Affinity DataIC50:  8nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245101((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(3-methylthio)p...)
Affinity DataIC50:  9nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245061((R)-3-{4-[3-(4-Cyano-3-trifluoromethylphenyl)-1-(4...)
Affinity DataIC50:  9nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244509((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(3-methoxy-5-tr...)
Affinity DataIC50:  9nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245057((R)-trans-3-{4-[1-(4-tert-Butyl-cyclohexyl)-3-(3-m...)
Affinity DataIC50:  10nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245060((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(4-trifluoromet...)
Affinity DataIC50:  12nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50:  12nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245100((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3-fluoro-...)
Affinity DataIC50:  13nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245059((R)-3-{4-[3-(3-Chlorophenyl)-1-(4-cyclohex-1-enylp...)
Affinity DataIC50:  14nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244508((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3-methoxy...)
Affinity DataIC50:  14nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244454((R/S)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3,5-dic...)
Affinity DataIC50:  14nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202041(CHEMBL375167 | trans-3-{4-[3-(3,5-Bis(trifluoromet...)
Affinity DataIC50:  16nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245062((R)-3-{4-[3-(3-tert-Butylphenyl)-1-(4-cyclohexylph...)
Affinity DataIC50:  18nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50171817(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50:  23nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50171817(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50:  23nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244505((R)-trans-3-{4-[1-(4-tert-Butylcyclohexyl)-3-(3,5-...)
Affinity DataIC50:  27nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50171817(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50:  28nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50:  36nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202060(3-{4-[1-(4-tert-Butylphenyl)-3-(4-trifluoromethoxy...)
Affinity DataIC50:  36nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202060(3-{4-[1-(4-tert-Butylphenyl)-3-(4-trifluoromethoxy...)
Affinity DataIC50:  38nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50171817(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50:  42nMAssay Description:Binding affinity to GIPR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244455((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3,5-dichl...)
Affinity DataIC50:  43nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244456((S)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3,5-dichl...)
Affinity DataIC50:  51nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245056((R/S)-3-{4-[1-(4-tert-Butylphenyl)-3-(4-trifluorom...)
Affinity DataIC50:  55nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50:  64nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245062((R)-3-{4-[3-(3-tert-Butylphenyl)-1-(4-cyclohexylph...)
Affinity DataIC50:  74nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244458((S)-trans-3-{4-[3-(3,5-Bis(trifluoromethyl)phenyl)...)
Affinity DataIC50:  82nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245099((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(2,2,4,4-t...)
Affinity DataIC50:  83nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244457((R)-trans-3-{4-[3-(3,5-Bis(trifluoromethyl)phenyl)...)
Affinity DataIC50:  87nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245098((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(3,5-dichloroph...)
Affinity DataIC50:  93nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202041(CHEMBL375167 | trans-3-{4-[3-(3,5-Bis(trifluoromet...)
Affinity DataIC50:  93nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245057((R)-trans-3-{4-[1-(4-tert-Butyl-cyclohexyl)-3-(3-m...)
Affinity DataIC50:  98nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244509((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(3-methoxy-5-tr...)
Affinity DataIC50:  145nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245058((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-phenyl-ure...)
Affinity DataIC50:  166nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245061((R)-3-{4-[3-(4-Cyano-3-trifluoromethylphenyl)-1-(4...)
Affinity DataIC50:  198nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244506((R)-3-{4-[3-(3-Bromophenyl)-1-(4-cyclohexylphenyl)...)
Affinity DataIC50:  216nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50:  216nMAssay Description:Binding affinity to GIPR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244505((R)-trans-3-{4-[1-(4-tert-Butylcyclohexyl)-3-(3,5-...)
Affinity DataIC50:  220nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245100((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3-fluoro-...)
Affinity DataIC50:  277nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244508((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3-methoxy...)
Affinity DataIC50:  279nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50245056((R/S)-3-{4-[1-(4-tert-Butylphenyl)-3-(4-trifluorom...)
Affinity DataIC50:  315nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244455((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3,5-dichl...)
Affinity DataIC50:  359nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244458((S)-trans-3-{4-[3-(3,5-Bis(trifluoromethyl)phenyl)...)
Affinity DataIC50:  373nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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